SCHEMBL5847324

SCHEMBL5847324

COc1ccc(-c2cc3c4c(c2C(C)(C)C)[C@@H]2CN(C(=O)O)CC[C@@H]2N4CC3)c(C=O)c1

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 2/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
FKBP1A P62942 8/20 0.33
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
ERN1 O75460 2/20 0.31
ABHD6 Q9BV23 1/20 0.31
ALDH1A1 P00352 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
RORC P51449 1/20 0.30
MTNR1B P49286 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847121 0.90 CCR3 (0.35) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5847619 0.89 CPS1 (0.37) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5847193 0.89 CCR3 (0.35) CCR3HTR2AHTR2CHTR2BFKBP1A
SCHEMBL5846973 0.87 CCR3 (0.34) CCR3HTR2AHTR2CHTR2BFKBP1A
SCHEMBL5847800 0.87 HTR2A (0.44) CCR3HTR2AHTR2CHTR2BESR1
SCHEMBL5410715 0.82 HTR2C (0.45) CCR3HTR2AHTR2CHTR2BFKBP1A
SCHEMBL5847913 0.81 ABCB1 (0.35) CCR3HTR2CFKBP1AALDH1A1MAPT
SCHEMBL5847854 0.81 HCRTR1 (0.36) CCR3HTR2AHTR2C
SCHEMBL5849715 0.80 DRD1 (0.37) CCR3HTR2AHTR2C
SCHEMBL5847475 0.79 S1PR1 (0.37) HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed