SCHEMBL5847475

SCHEMBL5847475

CC(C)Oc1ccc(-c2cc3c4c(c2C(C)(C)C)[C@@H]2CN(C(=O)O)CC[C@@H]2N4CC3)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.37
S1PR3 Q99500 1/20 0.37
HTR2A P28223 5/20 0.37
HTR2C P28335 2/20 0.37
HTR2B P41595 2/20 0.37
FFAR4 Q5NUL3 2/20 0.33
EPHX2 P34913 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5847800 0.92 HTR2A (0.44) HTR2AHTR2CHTR2BEPHX2
SCHEMBL5847306 0.90 HTR2A (0.36) HTR2AHTR2CHTR2BEPHX2
SCHEMBL5847107 0.86 SCD5 (0.37) HTR2AHTR2CHTR2BEPHX2DPP4
SCHEMBL5416030 0.84 HTR2A (0.52) S1PR1S1PR3HTR2AHTR2CHTR2B
SCHEMBL5846973 0.82 CCR3 (0.34) HTR2AHTR2CHTR2BDPP4
SCHEMBL5847619 0.82 CPS1 (0.37) HTR2AHTR2CHTR2B
SCHEMBL5847121 0.81 CCR3 (0.35) HTR2AHTR2CHTR2B
SCHEMBL5847193 0.80 CCR3 (0.35) HTR2AHTR2CHTR2BFFAR4
SCHEMBL5847324 0.79 CCR3 (0.34) HTR2AHTR2CHTR2B
SCHEMBL5410701 0.79 HTR2A (0.59) S1PR1S1PR3HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US claimed
US-7081455-B2 Substituted heterocycle fused gamma-carbolines BRISTOL-MYERS SQUIBB COMPANY (US) 2006-07-25 US disclosed