SCHEMBL5848640

SCHEMBL5848640

CC(C)(C)OC(=O)N1CCN(c2ncnc3sc([N+](=O)[O-])cc23)CC1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIT P10721 3/20 0.51
ALDH1A1 P00352 3/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
P2RY12 Q9H244 6/20 0.46
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 5/20 0.44
KCNH2 Q12809 1/20 0.43
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MET P08581 1/20 0.42
KMT2A Q03164 1/20 0.41
MAP4K4 O95819 1/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
FLT3 P36888 1/20 0.40
GBA1 P04062 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5851682 0.84 KIT (0.55) KITALDH1A1MAPTLMNAP2RY12
SCHEMBL7063655 0.84 ALDH1A1 (0.51) ALDH1A1MAPTLMNAP2RY12KDM4E
SCHEMBL7063657 0.84 ALDH1A1 (0.51) ALDH1A1MAPTLMNAP2RY12KDM4E
SCHEMBL5848798 0.83 KIT (0.57) KITALDH1A1MAPTP2RY12KDM4E
SCHEMBL5851315 0.83 KIT (0.54) KITALDH1A1MAPTP2RY12KDM4E
SCHEMBL5850542 0.83 KIT (0.54) KITALDH1A1MAPTP2RY12KDM4E
SCHEMBL5849579 0.82 KIT (0.53) KITALDH1A1MAPTLMNAP2RY12
SCHEMBL5850552 0.81 P2RY12 (0.68) ALDH1A1MAPTLMNAP2RY12KDM4E
SCHEMBL5849530 0.80 KIT (0.52) KITALDH1A1MAPTP2RY12KDM4E
SCHEMBL5849376 0.80 KIT (0.52) KITALDH1A1MAPTP2RY12KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7115741-B2 4-thieno[2,3-D]pyrimidin-4-YL piperazine compounds ALEXION PHARMACEUTICALS, INC. 2006-10-03 US disclosed
WO-2003022214-A2 PIPERAZINE AND HOMOPIPERAZINE COMPOUNDS MILLENNIUM PHARMACEUTICALS, INC. (US) 2003-03-20 WO disclosed