SCHEMBL5850463

SCHEMBL5850463

COC(=O)[C@H](Cc1ccc(NC(=O)C2CCN(C(=O)OC(C)(C)C)CC2)cc1)NC(=O)C1(N(C)S(=O)(=O)c2ccc(C)cc2)CCCC1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTPN2 P17706 1/20 0.46
PTPN1 P18031 1/20 0.46
PTPN6 P29350 1/20 0.46
ABL1 P00519 1/20 0.44
RIN1 Q13671 1/20 0.44
YAP1 P46937 1/20 0.43
KMT2A Q03164 3/20 0.42
MEN1 O00255 2/20 0.42
TRPV1 Q8NER1 1/20 0.42
P2RX7 Q99572 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
STS P08842 3/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
MMP13 P45452 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
EPHX2 P34913 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5852341 0.86 PTPN2 (0.48) PTPN2PTPN1PTPN6ABL1RIN1
SCHEMBL5851097 0.84 GHSR (0.39) KMT2AMEN1P2RX7
SCHEMBL5850976 0.79 ITGB1 (0.47) ALDH1A1LMNA
SCHEMBL5851039 0.78 ATM (0.55) ALDH1A1
SCHEMBL5850678 0.77 USP30 (0.44) KMT2AMEN1RAB9AALDH1A1LMNA
SCHEMBL5690604 0.77 ENPP2 (0.48) YAP1P2RX7NPC1RAB9AALDH1A1
SCHEMBL7409938 0.76 ATM (0.55) KMT2AALDH1A1
SCHEMBL5852314 0.76 ITGB1 (0.40) KMT2AALDH1A1GAA
SCHEMBL5850329 0.76 ITGB1 (0.41) P2RX7
SCHEMBL5851025 0.76 CA1 (0.45) KMT2ANPC1RAB9AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP claimed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US disclosed
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed