SCHEMBL5850585

SCHEMBL5850585

Cc1ccc(S(=O)(=O)N(C(=O)[C@@H]2CCCN2)[C@@](C)(Cc2ccc(OC(=O)N(C)C)cc2)C(=O)O)cc1

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.36
TAS2R14 Q9NYV8 5/20 0.35
SCN4A P35499 1/20 0.34
HTR2C P28335 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HTR2B P41595 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
ALOX5 P09917 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5850731 0.93 TAS2R14 (0.38) TAS2R14SCN4AHTR2CALDH1A1HTR2B
SCHEMBL5850625 0.92 PTGES (0.34) PTGESTAS2R14SCN4AHTR2CALDH1A1
SCHEMBL5852329 0.91 PTGES (0.33) PTGESTAS2R14SCN4AHTR2CALDH1A1
SCHEMBL5852564 0.86 NPY2R (0.38) ALDH1A1KMT2A
SCHEMBL5852560 0.85 CYP2C9 (0.45) ALDH1A1RAB9AKMT2A
SCHEMBL5852118 0.85 PSEN1 (0.35) TAS2R14SCN4AHTR2CALDH1A1HTR2B
SCHEMBL5850597 0.85 CYP2D6 (0.36) TAS2R14HTR2C
SCHEMBL5850614 0.84 PTGES (0.31) PTGESSCN4A
SCHEMBL5850526 0.79 ALDH1A1 (0.42) ALDH1A1LMNAMAPTRAB9AKMT2A
SCHEMBL5850848 0.78 L3MBTL1 (0.36) ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US claimed
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP claimed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed
US-7030114-B1 Compounds which inhibit leukocyte adhesion mediated by VLA-4 ELAN PHARMACEUTICALS, INC. (US) 2006-04-18 US disclosed
EP-0994895-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-04-26 EP disclosed
WO-1999006435-A1 DIPEPTIDE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed