SCHEMBL5859320

SCHEMBL5859320

COC1=C(OC)C(=O)C(c2ccc(C(=O)N3CCOCC3)c(-c3ccccc3)c2C)=C(C)C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.47
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 2/20 0.43
HPGD P15428 2/20 0.43
GAA P10253 1/20 0.43
ALOX15 P16050 1/20 0.43
CASP1 P29466 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TDP2 O95551 1/20 0.41
CNR1 P21554 1/20 0.41
EPHX1 P07099 1/20 0.41
APAF1 O14727 1/20 0.41
NPC1 O15118 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859070 0.90 SMN1; SMN2 (0.45) ALDH1A1HPGDLMNAHTTRAB9A
SCHEMBL5859035 0.89 HTT (0.41) TP53PDCD1CD274ALDH1A1KDM4E
SCHEMBL5862104 0.84 PLAUR (0.44) TP53ALDH1A1KDM4EHPGDGAA
SCHEMBL5860276 0.81 PDE4B (0.43) TP53ALDH1A1KDM4EHPGDALOX15
SCHEMBL5859955 0.79 CYP2C9 (0.43) TP53ALDH1A1HPGDHTTSMN1; SMN2
SCHEMBL5859916 0.77 RAB9A (0.49) ALDH1A1KDM4EHPGDGAAHSD17B10
SCHEMBL5859258 0.76 ALDH1A1 (0.40) TP53ALDH1A1KDM4EHPGDGAA
SCHEMBL5859907 0.75 RAB9A (0.49) ALDH1A1KDM4EHPGDHSD17B10CNR1
SCHEMBL5859144 0.74 EPHX1 (0.43) TP53PDCD1CD274ALDH1A1KDM4E
SCHEMBL5859316 0.74 CYP1A2 (0.42) PDCD1CD274ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122543-B2 Substituted benzoic acid derivatives having NF-κB inhibiting action DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2006-10-17 US disclosed
EP-1437339-A1 SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING NF-KAPPA B INHIBITING ACTIVITY Daiichi Suntory Pharma Co., Ltd. (JP) 2004-07-14 EP disclosed