SCHEMBL5860845

SCHEMBL5860845

COc1ccc(C(NC(=O)OC(C)(C)C)C(C)C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 2/20 0.51
PPARG P37231 1/20 0.48
PPARA Q07869 1/20 0.48
NPSR1 Q6W5P4 1/20 0.47
KEAP1 Q14145 7/20 0.44
NFE2L2 Q16236 7/20 0.44
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
PTGS2 P35354 3/20 0.40
PTGS1 P23219 2/20 0.40
AKR1C3 P42330 2/20 0.40
AKR1C2 P52895 2/20 0.40
CDC42 P60953 1/20 0.40
RAC1 P63000 1/20 0.40
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40
SLC22A6 Q4U2R8 1/20 0.40
MEN1 O00255 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6439138 0.86 ABCB1 (0.48) ABCB1PPARGPPARANPSR1CTSS
SCHEMBL26647713 0.86 CTSS (0.47) KEAP1NFE2L2CTSSCTSKCYP1A2
SCHEMBL12732987 0.86 ABCB1 (0.53) ABCB1PPARGPPARANPSR1CTSS
SCHEMBL1573516 0.86 KEAP1 (0.51) PPARGPPARAKEAP1NFE2L2CTSS
SCHEMBL15165758 0.86 KEAP1 (0.51) PPARGPPARAKEAP1NFE2L2CTSS
SCHEMBL5862225 0.86 KEAP1 (0.51) PPARGPPARAKEAP1NFE2L2CTSS
SCHEMBL23205818 0.85 PPARG (0.47) PPARGPPARAKEAP1NFE2L2CTSS
SCHEMBL12732988 0.85 ABCB1 (0.52) ABCB1PPARGPPARANPSR1CTSS
SCHEMBL20521905 0.85 PPARG (0.47) PPARGPPARAKEAP1NFE2L2CTSS
SCHEMBL6513379 0.85 KEAP1 (0.42) ABCB1PPARGPPARAKEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7041667-B1 CCR5 modulators PFIZER, INC. (US) 2006-05-09 US disclosed
EP-1013276-A1 Aminoazacycloalkanes as CCR5 modulators PFIZER INC. (US) 2000-06-28 EP disclosed