SCHEMBL586141

SCHEMBL586141

Cc1ccc(Nc2c(F)cccc2Cl)c(C(CCc2ccc(N3C(O)c4ccccc4C3O)cc2)C(=O)O)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.49
PTGS1 P23219 3/20 0.49
ABCB11 O95342 1/20 0.49
PPARG P37231 1/20 0.49
NR1I3 Q14994 1/20 0.49
CXCL8 P10145 1/20 0.35
PTGES O14684 1/20 0.33
MAPK8 P45983 2/20 0.33
MAPK9 P45984 2/20 0.33
MAPK10 P53779 2/20 0.33
MAPK14 Q16539 2/20 0.33
MT-CO2 P00403 1/20 0.33
CRHR1 P34998 1/20 0.32
RAB9A P51151 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CSNK1E P49674 1/20 0.31
DDR1 Q08345 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL577459 0.80 PTGS2 (0.54) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL577022 0.80 PTGS2 (0.45) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL7131340 0.76 PTGS2 (0.67) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL585080 0.75 CXCL8 (0.48) PTGS2PTGS1ABCB11NR1I3CXCL8
SCHEMBL27595572 0.73 PTGS2 (0.64) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL576775 0.73 PTGS2 (0.65) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL586377 0.70 CXCL8 (0.47) PTGS2PTGS1ABCB11NR1I3CXCL8
SCHEMBL7129516 0.69 PTGS2 (0.53) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL7122501 0.69 PTGS2 (0.64) PTGS2PTGS1ABCB11PPARGNR1I3
Lumiracoxib SCHEMBL4479 0.67 PTGS2 (1.00) PTGS2PTGS1ABCB11PPARGNR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2418200-A1 PHTHALIMIDE DERIVATIVES OF NON-STEROIDAL ANTI-INFLAMMATORY COMPOUNDS AND/OR TNF- MODULATORS, METHOD FOR PRODUCING SAME, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND USES THEREOF FOR THE TREATMENT OF INFLAMMATORY DISEASES EMS S. A. (BR) 2012-02-15 EP claimed