SCHEMBL5861503

SCHEMBL5861503

Nc1nc2c(ncn2[C@@H]2O[C@H](C(O)OP(=O)(O)O)[C@H](O)[C@H]2O)c(=O)[nH]1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.60
TGM2 P21980 1/20 0.56
IMPDH2 P12268 6/20 0.54
HINT1 P49773 1/20 0.53
STING1 Q86WV6 2/20 0.52
PDE3B Q13370 1/20 0.52
PDE3A Q14432 1/20 0.52
TAAR1 Q96RJ0 1/20 0.51
KRAS P01116 4/20 0.51
IMPDH1 P20839 2/20 0.50
GSK3A P49840 2/20 0.50
RPS6KA3 P51812 2/20 0.50
MAPK14 Q16539 2/20 0.50
FUT5 Q11128 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4081026 1.00 NT5E (0.60) NT5ETGM2IMPDH2HINT1STING1
Guanosine SCHEMBL2447866 0.93 NT5E (0.62) NT5ETGM2IMPDH2HINT1KRAS
SCHEMBL9124928 0.92 NT5E (0.53) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL407394 0.90 NT5E (0.59) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL1527362 0.90 NT5E (0.59) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL19183426 0.88 NT5E (0.57) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL22636005 0.87 NT5E (0.62) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL22498538 0.87 NT5E (0.62) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL4651242 0.87 NT5E (0.56) NT5ETGM2IMPDH2HINT1STING1
SCHEMBL30867115 0.87 NT5E (0.53) NT5ETGM2IMPDH2HINT1STING1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7122572-B2 For use in Hydrogen Bonding Liquid Chromatography, environmental remediation by removal of undesired ions or neutral molecules, removal of phosphate for kidney dialysis, drug delivery, separation BOARD OF REGENTS, UNIVERSITY OF TEXAS SYSTEM (US) 2006-10-17 US disclosed
US-7041819-B2 Halogenated calixpyrroles and uses thereof BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2006-05-09 US disclosed
US-6984734-B2 Cyclo[n]pyrroles and methods thereto BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2006-01-10 US disclosed
US-20030229131-A1 Cyclo[n]pyrroles and methods thereto BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2003-12-11 US disclosed
WO-2003072581-A1 CYCLO[N]PYRROLES AND METHODS THERETO BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2003-09-04 WO disclosed
WO-2003018548-A2 HALOGENATED CALIXPYRROLES, CALIXPYRIDINOPYRROLES AND CALIXPYRIDINES, AND USES THEREOF BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 2003-03-06 WO disclosed
US-20020115566-A1 Halogenated calixpyrroles, calixpyridinopyrroles and calixpyridines, and uses thereof BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM 2002-08-22 US disclosed
US-20020026047-A1 Calixpyrroles, calixpyridinopyrroles, and calixpyridines BOARD OF REGENTS, THE 2002-02-28 US disclosed
US-6262257-B1 SELECTIVE ION- AND NEUTRAL MOLECULE-BINDING AGENTS FORMING SUPRAMOLECULAR ENSEMBLES, AND ION- AND NEUTRAL MOLECULE-SEPARATION AGENTS BOARD OF REGENTS, UNIVERSITY OF TEXAS SYSTEM 2001-07-17 US disclosed
EP-0891364-A1 CALIXPYRROLES, CALIXPYRIDINOPYRROLES AND CALIXPYRIDINES THE BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1999-01-20 EP disclosed
US-5808059-A CHROMATOGRAPHY; ELECTROPHORESIS BOARD OF REGENTS, UNIVERSITY OF TEXAS SYSTEM (US) 1998-09-15 US disclosed
US-5744302-A USING A PORPHYRIN; COMPLEXING BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1998-04-28 US disclosed
WO-1997037995-A1 CALIXPYRROLES, CALIXPYRIDINOPYRROLES AND CALIXPYRIDINES BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1997-10-16 WO disclosed
US-5672490-A PROMOTING THE SPLITTING DNA BY MIXING WITH A SAPPHYRIN-EDTA CONJUGATE COMPOUND THE UNIVERSITY OF TEXAS BOARD OF REGENTS (US) 1997-09-30 US disclosed
US-5530123-A ANTIVIRAL AND CHEMOTHERAPEUTICAL AGENT FOR CANCER BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1996-06-25 US disclosed
US-5457195-A Sapphyrin derivatives and conjugates BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1995-10-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229131-A1 Cyclo[n]pyrroles and methods thereto PPOX, QPCT, PPIE NT5E 706/4885TGM2 3279/4885IMPDH2 1607/4885
US-20020115566-A1 Halogenated calixpyrroles, calixpyridinopyrroles and calixpyridines, and uses thereof CALD1, CALU, CLASP1 NT5E 3680/4885TGM2 3797/4885IMPDH2 3386/4885
US-20020026047-A1 Calixpyrroles, calixpyridinopyrroles, and calixpyridines CALD1, DAP3, CALR NT5E 3281/4885TGM2 2752/4885IMPDH2 3016/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.