SCHEMBL5863083

SCHEMBL5863083

CN(C)CCNC(=O)c1ccc(-c2ccccc2CSCCOc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
HPGD P15428 2/20 0.46
POLB P06746 1/20 0.46
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
ALOX5 P09917 1/20 0.45
FYN P06241 1/20 0.45
RAD52 P43351 1/20 0.45
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
GPR55 Q9Y2T6 1/20 0.43
MAPT P10636 1/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
CACNA1H O95180 1/20 0.42
CACNA1B Q00975 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5863100 0.94 FYN (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL5863072 0.93 NPC1 (0.45) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
Oxalic Acid SCHEMBL5863143 0.88 FYN (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
Oxalic Acid SCHEMBL5863159 0.85 ALDH1A1 (0.51) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
Oxalic Acid SCHEMBL5863050 0.84 KCNA5 (0.43) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
Oxalic Acid SCHEMBL5863262 0.83 FYN (0.46) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL5863380 0.83 ROCK2 (0.50) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
Oxalic Acid SCHEMBL5863102 0.82 KDR (0.44) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD
SCHEMBL6252851 0.82 KDM4E (0.43) ALDH1A1SMN1; SMN2KMT2AMAPTCD274
SCHEMBL5641530 0.81 ALDH1A1 (0.47) ALDH1A1NPC1RAB9ASMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7132456-B2 MCH receptor antagonists ELI LILLY AND COMPANY (US) 2006-11-07 US disclosed
US-20060052449-A1 Novel mch receptor antagonists ELI LILLY AND COMPANY 2006-03-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060052449-A1 Novel mch receptor antagonists MCHR1, MCHR2, MC1R ALDH1A1 1500/4885NPC1 698/4885RAB9A 996/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.