SCHEMBL5863128

SCHEMBL5863128

O=Cc1nn2c(Cl)ccc2c(=O)n1Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.42
ALDH1A1 P00352 5/20 0.40
NPSR1 Q6W5P4 2/20 0.40
LMNA P02545 1/20 0.40
CFTR P13569 1/20 0.40
HPGD P15428 2/20 0.39
KDM4E B2RXH2 2/20 0.39
KDM4A O75164 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
P2RX4 Q99571 1/20 0.38
ADORA1 P30542 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
FGFR1 P11362 1/20 0.38
FGFR3 P22607 1/20 0.38
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
PIK3CA P42336 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5863491 0.83 KIF11 (0.42) KIF11ALDH1A1NPSR1CFTRHPGD
SCHEMBL5863538 0.81 KIF11 (0.48) KIF11ALDH1A1NPSR1LMNACFTR
SCHEMBL5863800 0.73 KIF11 (0.55) KIF11ALDH1A1NPSR1CFTRHPGD
SCHEMBL5863079 0.72 KIF11 (0.44) KIF11ALDH1A1NPSR1LMNAHPGD
SCHEMBL5863209 0.72 KIF11 (0.56) KIF11ALDH1A1NPSR1LMNACFTR
SCHEMBL5863442 0.72 KIF11 (0.56) KIF11ALDH1A1NPSR1CFTRHPGD
SCHEMBL2084701 0.65 VDR (0.72) ALDH1A1NPSR1LMNACFTRHPGD
SCHEMBL8985073 0.62 GSK3B (0.67) ALDH1A1LMNAHPGDKDM4EL3MBTL1
SCHEMBL16818583 0.60 TDP1 (0.46) ALDH1A1NPSR1LMNACFTRKDM4E
SCHEMBL96124 0.60 SRC (0.51) ALDH1A1NPSR1LMNAHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030118-B2 Pyrrolotriazinone compounds and their use to treat diseases BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-18 US disclosed
US-20030232832-A1 Nitrogen compounds such as N-(3-Aminopropyl)-N-(1-(3-benzyl-4 -oxo-3,4-dihydropyrrolo(2,1-f)(1,2,4)-triazine-2-yl)-propyl)-4 -methylbenzamide, trifluoroacetic acid salt, used as anticarcinogenic or antiproliferative agents BRISTOL-MYERS SQUIBB COMPANY 2003-12-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030232832-A1 Nitrogen compounds such as N-(3-Aminopropyl)-N-(1-(3-benzyl-4 -oxo-3,4-dihydropyrrolo(2,1-f)(1,2,4)-triazine-2-yl)-propyl)-4 -methylbenzamide, trifluoroacetic acid salt, used as anticarcinogenic or antiproliferative agents CCNB1, NUMA1, CCNA1 KIF11 858/4885ALDH1A1 1027/4885NPSR1 2690/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.