SCHEMBL5863209

SCHEMBL5863209

O=c1c2ccc(Cl)n2nc(C(O)C2CC2)n1Cc1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.56
TDP1 Q9NUW8 1/20 0.35
PIK3CA P42336 1/20 0.35
CFTR P13569 1/20 0.35
ALDH1A1 P00352 3/20 0.34
HTT P42858 2/20 0.34
HPGD P15428 2/20 0.34
KDM4E B2RXH2 2/20 0.34
KDM4A O75164 1/20 0.34
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 1/20 0.34
PDE1A P54750 1/20 0.34
PDE1B Q01064 1/20 0.34
PDE1C Q14123 1/20 0.34
CASR P41180 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5863800 0.87 KIF11 (0.55) KIF11TDP1PIK3CACFTRALDH1A1
SCHEMBL5863442 0.86 KIF11 (0.56) KIF11TDP1PIK3CACFTRALDH1A1
SCHEMBL5863057 0.76 KIF11 (0.56) KIF11
SCHEMBL5863538 0.74 KIF11 (0.48) KIF11TDP1PIK3CACFTRALDH1A1
SCHEMBL5863128 0.72 KIF11 (0.42) KIF11TDP1PIK3CACFTRALDH1A1
SCHEMBL4251309 0.68 HPGD (0.41) KIF11ALDH1A1HTTHPGDKDM4E
SCHEMBL5863491 0.67 KIF11 (0.42) KIF11TDP1PIK3CACFTRALDH1A1
SCHEMBL4246757 0.65 HPGD (0.41) KIF11ALDH1A1HTTHPGDKDM4E
SCHEMBL31315686 0.64 CFTR (0.51) TDP1CFTRALDH1A1NPSR1
SCHEMBL5863432 0.64 KIF11 (0.55) KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7030118-B2 Pyrrolotriazinone compounds and their use to treat diseases BRISTOL-MYERS SQUIBB COMPANY (US) 2006-04-18 US disclosed
US-20030232832-A1 Nitrogen compounds such as N-(3-Aminopropyl)-N-(1-(3-benzyl-4 -oxo-3,4-dihydropyrrolo(2,1-f)(1,2,4)-triazine-2-yl)-propyl)-4 -methylbenzamide, trifluoroacetic acid salt, used as anticarcinogenic or antiproliferative agents BRISTOL-MYERS SQUIBB COMPANY 2003-12-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030232832-A1 Nitrogen compounds such as N-(3-Aminopropyl)-N-(1-(3-benzyl-4 -oxo-3,4-dihydropyrrolo(2,1-f)(1,2,4)-triazine-2-yl)-propyl)-4 -methylbenzamide, trifluoroacetic acid salt, used as anticarcinogenic or antiproliferative agents CCNB1, NUMA1, CCNA1 KIF11 858/4885TDP1 381/4885PIK3CA 1240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.