SCHEMBL586674

SCHEMBL586674

COC(=O)C1CCN(C(=O)OC)C(c2ccc(C(F)(F)F)cc2)C1.COC(=O)N1CCC(C(=O)O)CC1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.44
TDP1 Q9NUW8 3/20 0.42
MAPK1 P28482 2/20 0.42
ALDH1A1 P00352 2/20 0.42
GAA P10253 2/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 2/20 0.40
CYP3A4 P08684 2/20 0.37
PSEN1 P49768 1/20 0.36
PSEN2 P49810 1/20 0.36
APH1B Q8WW43 1/20 0.36
NCSTN Q92542 1/20 0.36
APH1A Q96BI3 1/20 0.36
PSENEN Q9NZ42 1/20 0.36
SLC6A9 P48067 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL586946 0.96 TDP1 (0.45) NOTUMTDP1MAPK1ALDH1A1GAA
SCHEMBL582132 0.96 NOTUM (0.47) NOTUMTDP1MAPK1ALDH1A1GAA
SCHEMBL5258300 0.89 TDP1 (0.45) NOTUMTDP1MAPK1ALDH1A1GAA
SCHEMBL587349 0.88 MMP1 (0.41) NOTUM
SCHEMBL586941 0.88 NOTUM (0.45) NOTUMTDP1ALDH1A1GAAKDM4E
SCHEMBL2859600 0.87 MAPT (0.43) TDP1MAPK1ALDH1A1GAAKDM4E
SCHEMBL587057 0.85 TACR1 (0.40) NOTUMTDP1MAPT
SCHEMBL587433 0.85 SMN1; SMN2 (0.44) NOTUMMAPT
SCHEMBL586744 0.85 SLC6A2 (0.46) TDP1ALDH1A1KDM4EMAPTCYP3A4
SCHEMBL581263 0.85 SLC6A2 (0.41) TDP1ALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed