SCHEMBL587092

SCHEMBL587092

COC(=O)C1CCN(C(=O)OC)C(C(F)F)C1.COC(=O)N1CCC(C(=O)O)CC1C(F)F

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.37
SMN1; SMN2 Q16637 3/20 0.35
ALDH1A1 P00352 5/20 0.34
GAA P10253 2/20 0.33
POLB P06746 1/20 0.33
TSHR P16473 2/20 0.33
MAPT P10636 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
OPRK1 P41145 1/20 0.31
KDM4E B2RXH2 1/20 0.31
BTK Q06187 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581073 0.94 TSHR (0.36) TP53GAATSHRRAB9AHSD17B10
SCHEMBL587449 0.94 TP53 (0.41) TP53SMN1; SMN2ALDH1A1GAAPOLB
SCHEMBL582298 0.78 NOTUM (0.32) TSHRKDM4ELMNA
SCHEMBL581244 0.74 GAA (0.36) ALDH1A1GAATSHRMAPTKDM4E
SCHEMBL3074935 0.74 GAA (0.36) ALDH1A1GAATSHRMAPTKDM4E
SCHEMBL580903 0.74 GAA (0.36) ALDH1A1GAATSHRMAPTKDM4E
SCHEMBL582099 0.73 TSHR (0.48) TP53SMN1; SMN2GAATSHRMAPT
SCHEMBL587349 0.73 MMP1 (0.41)
SCHEMBL587629 0.72 ALDH1A1 (0.34) SMN1; SMN2ALDH1A1MAPTNPSR1NPC1
SCHEMBL587099 0.72 ALDH1A1 (0.34) TP53SMN1; SMN2ALDH1A1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed