SCHEMBL5872354

SCHEMBL5872354

CC(C)CC1NC(=O)OC1(c1ccccc1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
PAX8 Q06710 1/20 0.35
ATM Q13315 1/20 0.33
CCR5 P51681 4/20 0.32
MMP3 P08254 2/20 0.32
CASP1 P29466 2/20 0.32
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
HSD11B1 P28845 1/20 0.31
CHRM2 P08172 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM1 P11229 1/20 0.31
CHRM3 P20309 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
ELANE P08246 1/20 0.31
CCKBR P32239 1/20 0.30
MEN1 O00255 1/20 0.30
CYP1A2 P05177 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872352 1.00 GAA (0.35) GAAHTTPAX8ATMCCR5
SCHEMBL6941289 0.80 TSHR (0.34) MMP3MMP2MMP9MEN1CYP1A2
SCHEMBL5872468 0.78 HDAC8 (0.36) GAAHTTCYP1A2POLBTSHR
SCHEMBL5872462 0.78 HDAC8 (0.36) GAAHTTCYP1A2POLBTSHR
SCHEMBL7780090 0.78 MMP2 (0.38) MMP3MMP2MMP9MEN1CYP1A2
SCHEMBL2077742 0.76 ATM (0.35) ATMMMP2MMP9HSD11B1CYP1A2
SCHEMBL2513974 0.76 ATM (0.35) ATMMMP2MMP9HSD11B1CYP1A2
SCHEMBL2077738 0.76 ATM (0.35) ATMMMP2MMP9HSD11B1CYP1A2
SCHEMBL5872252 0.75 CYP1A2 (0.36) GAAATMHSD11B1ELANEMEN1
SCHEMBL5872329 0.75 CYP1A2 (0.36) GAAATMHSD11B1ELANEMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2943475-B1 PROCESS FOR THE PREPARATION OF A FLUOROLACTON DERIVATIVE GILEAD PHARMASSET LLC (US) 2017-10-25 EP disclosed
US-7126028-B1 Process for preparing chiral compounds THE UNIVERSITY COURT OF THE UNIVERSITY OF ST. ANDREWS (GB) 2006-10-24 US disclosed
EP-1135349-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2001-09-26 EP disclosed
WO-2000034210-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2000-06-15 WO disclosed