SCHEMBL5872468

SCHEMBL5872468

O=C1NC(Cc2ccccc2)C(c2ccccc2)(c2ccccc2)O1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.36
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
TLR9 Q9NR96 1/20 0.36
CA2 P00918 1/20 0.36
MAOB P27338 1/20 0.36
EP300 Q09472 1/20 0.35
CTRB1 P17538 1/20 0.34
GAA P10253 2/20 0.34
POLB P06746 1/20 0.34
CES2 O00748 1/20 0.34
TSHR P16473 1/20 0.34
HTT P42858 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872462 1.00 HDAC8 (0.36) HDAC8DDB1CRBNTLR9CA2
SCHEMBL31403360 1.00 HDAC8 (0.36) HDAC8DDB1CRBNTLR9CA2
SCHEMBL6941289 0.79 TSHR (0.34) POLBTSHRCYP1A2CYP2C19KMT2A
SCHEMBL2369273 0.79 LMNA (0.42) HDAC8DDB1CRBNTLR9CA2
SCHEMBL531694 0.79 LMNA (0.42) HDAC8DDB1CRBNTLR9CA2
SCHEMBL531693 0.79 LMNA (0.42) HDAC8DDB1CRBNTLR9CA2
SCHEMBL5872352 0.78 GAA (0.35) GAAPOLBTSHRHTTCYP1A2
SCHEMBL5872354 0.78 GAA (0.35) GAAPOLBTSHRHTTCYP1A2
SCHEMBL7780090 0.77 MMP2 (0.38) CYP1A2CYP3A4CYP2C19KMT2A
SCHEMBL13949518 0.74 LMNA (0.38) HDAC8DDB1CRBNTLR9CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7126028-B1 Process for preparing chiral compounds THE UNIVERSITY COURT OF THE UNIVERSITY OF ST. ANDREWS (GB) 2006-10-24 US disclosed
EP-1135349-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2001-09-26 EP disclosed
WO-2000034210-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2000-06-15 WO disclosed