SCHEMBL5872368

SCHEMBL5872368

CN[C@@H](C(C)C)C(F)(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 3/20 0.40
TSHR P16473 3/20 0.39
ALDH1A1 P00352 1/20 0.39
TAAR1 Q96RJ0 2/20 0.35
SLC18A2 Q05940 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
CYP2D6 P10635 3/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C19 P33261 2/20 0.34
CHRM2 P08172 1/20 0.34
ADRA1A P35348 1/20 0.34
RGS12 O14924 1/20 0.34
GLA P06280 1/20 0.34
CYP2C9 P11712 1/20 0.34
PKM P14618 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
ADRA2C P18825 1/20 0.34
NFKB1 P19838 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14233970 0.78 KCNN4 (0.41) KCNN4TSHRALDH1A1TAAR1SLC18A2
SCHEMBL19448773 0.73 ALDH1A1 (0.50) KCNN4TSHRALDH1A1TAAR1CYP2D6
SCHEMBL1167957 0.70 ALDH1A1 (0.46) KCNN4TSHRALDH1A1TAAR1SIGMAR1
Trifluoromethylbenzene SCHEMBL1768875 0.66 TSHR (0.78) KCNN4TSHRALDH1A1SIGMAR1CYP2D6
SCHEMBL10419000 0.66 TSHR (0.52) KCNN4TSHRALDH1A1CYP1A2PTPN1
SCHEMBL17922094 0.65
SCHEMBL17922085 0.65
SCHEMBL14268034 0.65
SCHEMBL12356881 0.64 ALDH1A1 (0.50) KCNN4TSHRALDH1A1TAAR1CYP2D6
SCHEMBL3879900 0.64 KCNN4 (0.56) KCNN4TSHRALDH1A1TAAR1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1135349-B1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIV ST ANDREWS (GB) 2005-04-06 EP claimed
US-7126028-B1 Process for preparing chiral compounds THE UNIVERSITY COURT OF THE UNIVERSITY OF ST. ANDREWS (GB) 2006-10-24 US disclosed
EP-1135349-B1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIV ST ANDREWS (GB) 2005-04-06 EP disclosed
EP-1135349-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2001-09-26 EP disclosed
WO-2000034210-A1 PROCESS FOR PREPARING CHIRAL COMPOUNDS UNIVERSITY OF DURHAM (GB) 2000-06-15 WO disclosed