SCHEMBL5872381

SCHEMBL5872381

N#CCN1CCC[C@@H]1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.39
POLB P06746 1/20 0.39
SPHK1 Q9NYA1 1/20 0.38
SCN3A Q9NY46 1/20 0.36
DPP4 P27487 4/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
LMNA P02545 1/20 0.36
CD274 Q9NZQ7 1/20 0.34
HRH3 Q9Y5N1 4/20 0.33
GRM2 Q14416 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5872372 0.95 AR (0.35) ARPOLBSPHK1SCN3ADPP4
SCHEMBL2224080 0.84 CYP1A2 (0.40) LMNA
SCHEMBL14940944 0.84 POLB (0.39) ARPOLBSPHK1SCN3ADPP4
SCHEMBL2224084 0.84 CYP1A2 (0.40) LMNA
SCHEMBL6020379 0.80 ALDH1A1 (0.37) LMNA
SCHEMBL6020376 0.80 F2 (0.37) DPP4HSD11B1
SCHEMBL2224603 0.78 LTA4H (0.43) POLB
SCHEMBL2224182 0.78 LTA4H (0.43) POLB
SCHEMBL12201786 0.77 POLB (0.42) ARPOLBSPHK1SCN3ADPP4
SCHEMBL943039 0.77 POLB (0.42) ARPOLBSPHK1SCN3ADPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7012075-B2 Cathepsin cysteine protease inhibitors MERCK & CO., INC. (US) 2006-03-14 US disclosed