SCHEMBL5876953

SCHEMBL5876953

Cc1ccc(-c2nc3ccc(C)cc3c(=O)n2CC2CCCC(CN)C2)cc1

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.50
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP2D6 P10635 4/20 0.43
HTR2C P28335 1/20 0.43
GHSR Q92847 4/20 0.42
CYP3A4 P08684 1/20 0.42
KCNH2 Q12809 1/20 0.42
AVPR1B P47901 4/20 0.41
RORC P51449 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877732 0.95 ABCC1 (0.52) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL5877626 0.95 ABCC1 (0.52) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL5877963 0.92 ALDH1A1 (0.47) ABCC1MEN1KMT2AALDH1A1GHSR
SCHEMBL5877579 0.92 ABCC1 (0.46) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL5877998 0.92 MEN1 (0.53) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL5877811 0.92 ABCC1 (0.46) ABCC1KMT2ACYP2D6HTR2CGHSR
SCHEMBL5877870 0.90 ABCC1 (0.48) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL5877563 0.90 F11 (0.50) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL5877265 0.90 ABCC1 (0.44) ABCC1MEN1KMT2AALDH1A1CYP2D6
SCHEMBL7492616 0.89 ABCC1 (0.42) ABCC1MEN1KMT2AALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed