SCHEMBL5877963

SCHEMBL5877963

COc1ccc(-c2nc3ccc(C)cc3c(=O)n2CC2CCCC(CN)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.47
KDM4E B2RXH2 4/20 0.47
MAPT P10636 3/20 0.47
HPGD P15428 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 2/20 0.47
MAPK1 P28482 1/20 0.47
F11 P03951 1/20 0.46
ABCC1 P33527 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
ADRA1A P35348 1/20 0.44
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
AVPR1B P47901 3/20 0.42
CYP1A2 P05177 1/20 0.41
POLB P06746 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
GHSR Q92847 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877563 0.94 F11 (0.50) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL5876981 0.94 F11 (0.52) ALDH1A1KDM4EMAPTHPGDLMNA
SCHEMBL5877265 0.94 ABCC1 (0.44) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL5876985 0.92 CRHR1 (0.44) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL5876953 0.92 ABCC1 (0.50) ALDH1A1SMN1; SMN2ABCC1MEN1KMT2A
SCHEMBL5877561 0.91 CYP2D6 (0.46) F11ABCC1MEN1KMT2AADRA1A
SCHEMBL5877862 0.90 AVPR1B (0.46) MAPTLMNAABCC1AVPR1BNPSR1
SCHEMBL5877069 0.90 F11 (0.49) F11ABCC1MEN1KMT2AADRA1A
SCHEMBL5877978 0.90 AVPR1B (0.49) F11ABCC1MEN1KMT2AADRA1A
SCHEMBL5877732 0.89 ABCC1 (0.52) ALDH1A1ABCC1MEN1KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed