SCHEMBL5876985

SCHEMBL5876985

COc1ccc(-c2ccc(-c3nc4ccc(C)cc4c(=O)n3CC3CCCC(CN)C3)cc2)c(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.44
F11 P03951 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 2/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ADRA1A P35348 1/20 0.42
KCNH2 Q12809 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
GRIN1 Q05586 1/20 0.42
GRIN2B Q13224 1/20 0.42
ABCC1 P33527 1/20 0.41
GHSR Q92847 2/20 0.40
P2RX3 P56373 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PTGER4 P35408 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5877807 0.96 F11 (0.47) CRHR1F11ADRA1AKCNH2HRH3
SCHEMBL5877963 0.92 ALDH1A1 (0.47) F11ALDH1A1MAPTHPGDMAPK1
SCHEMBL5877425 0.92 CYP2D6 (0.43) CRHR1F11ADRA1AKCNH2HRH3
SCHEMBL5877906 0.91 ABCC1 (0.52) CRHR1ALDH1A1MAPTHPGDMAPK1
SCHEMBL5877563 0.90 F11 (0.50) F11ALDH1A1MAPTHPGDMAPK1
SCHEMBL5877936 0.89 CRHR1 (0.41) CRHR1F11LMNAADRA1AKCNH2
SCHEMBL5876981 0.89 F11 (0.52) F11ALDH1A1MAPTHPGDMAPK1
SCHEMBL5877265 0.88 ABCC1 (0.44) F11ALDH1A1MAPTHPGDMAPK1
SCHEMBL5878313 0.87 PDE4B (0.43) ALDH1A1MAPTHPGDMAPK1KDM4E
SCHEMBL5877717 0.87 EGFR (0.44) CRHR1MAPK1KCNH2HRH3GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7060706-B1 Quinazolinones 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 2006-06-13 US disclosed
EP-1216233-A1 QUINAZOLINONES MERCK PATENT GmbH (DE) 2002-06-26 EP disclosed
WO-2001023364-A1 QUINAZOLINONES MERCK PATENT GMBH (DE) 2001-04-05 WO disclosed