SCHEMBL588118

SCHEMBL588118

Cc1nc(F)c(F)c(C(=O)O)c1C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.39
TAS1R3 Q7RTX0 4/20 0.35
TAS1R1 Q7RTX1 3/20 0.35
TAS1R2 Q8TE23 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
HIF1A Q16665 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KMO O15229 1/20 0.32
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
TYK2 P29597 1/20 0.31
JAK3 P52333 1/20 0.31
LIPE Q05469 2/20 0.31
MAT2A P31153 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL588119 0.80 DHODH (0.42) DHODHTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL18781916 0.78 KMO (0.37) DHODHTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL15022565 0.73 HCAR2 (0.35) DHODHSMN1; SMN2KDM4EHTTKMT2A
SCHEMBL14989167 0.70 KMO (0.41) SMN1; SMN2KDM4EGLAHTTKMT2A
SCHEMBL17323560 0.70 DHODH (0.36) DHODHTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL1264771 0.68 ACMSD (0.38) SMN1; SMN2KDM4EGLAHTTKMT2A
SCHEMBL2311682 0.67 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2SMN1; SMN2KMT2A
SCHEMBL28844067 0.67 TAS1R3 (0.44) DHODHTAS1R3TAS1R1TAS1R2SMN1; SMN2
SCHEMBL14989298 0.67 KMO (0.39) DHODHSMN1; SMN2KDM4EGLAHTT
SCHEMBL14989223 0.67 KMO (0.39) DHODHSMN1; SMN2KDM4EGLAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417131-A1 ISOXAZOL-3(2H)-ONE ANALOGS AS THERAPEUTIC AGENTS AstraZeneca AB (SE) 2012-02-15 EP disclosed
WO-2010117323-A1 METHOD AND APPARATUS FOR PRODUCING HEAT ENERGY AND CARBON DIOXIDE ASTRAZENECA AB (SE) 2010-10-14 WO disclosed