SCHEMBL588221

SCHEMBL588221

BrCc1ccc(-c2ccccc2)c(-c2nnnn2C(c2ccccc2)(c2ccccc2)c2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.44
AGTR2 P50052 1/20 0.44
AGT P01019 2/20 0.36
POLB P06746 2/20 0.34
ALDH1A1 P00352 2/20 0.32
HTT P42858 2/20 0.32
TACR1 P25103 2/20 0.32
P2RX7 Q99572 2/20 0.32
HDAC6 Q9UBN7 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
TSHR P16473 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
DRD4 P21917 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29931185 1.00 AGTR1 (0.44) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL27873329 0.91 AGTR1 (0.44) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL29931122 0.89 AGTR1 (0.44) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL27586872 0.89 AGTR1 (0.44) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL796 0.89 AGTR1 (0.50) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL29404889 0.89 AGTR1 (0.50) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL27631745 0.88 AGTR1 (0.44) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL8698703 0.83 AGTR1 (0.47) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL2053236 0.82 AGTR1 (0.44) AGTR1AGTR2AGTPOLBALDH1A1
SCHEMBL7196989 0.82 AGTR1 (0.41) AGTR1AGTR2POLBALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119039279-A Synthesis process of trityl olmesartan medoxomil 浙江华洋药业有限公司 2024-11-29 CN claimed
CN-113666881-A Synthesis method of mutagenic azide impurities in tetrazole sartan bulk drugs 河南华商药业有限公司 2021-11-19 CN claimed
CN-101328167-B Preparation method of losartan BEIJING SECOND PHARMACEUTICAL CO LTD 2012-04-25 CN claimed
EP-1753746-B8 NOVEL PYRROLE DERIVATIVES WITH ANGIOTENSIN II ANTAGONIST ACTIVITY ROTTAPHARM SPA (IT) 2012-02-15 EP claimed
EP-2049527-A2 PREPARATION OF IRBESARTAN Krka Tovarna Zdravil, D.D., Novo Mesto (SI) 2009-04-22 EP claimed
EP-1753746-A2 NOVEL PYRROLE DERIVATIVES WITH ANGIOTENSIN II ANTAGONIST ACTIVITY ROTTAPHARM S.P.A. (IT) 2007-02-21 EP claimed
WO-2006073376-A2 PREPARATION OF IRBESARTAN KRKA, TOVARNA ZDRAVIL, D.D., NOVO MESTO (SI) 2006-07-13 WO claimed
WO-2005105789-A2 NOVEL PYRROLE DERIVATIVES WITH ANGIOTENSIN II ANTAGONIST ACTIVITY ROTTAPHARM S.P.A. (IT) 2005-11-10 WO claimed
CN-119039279-A Synthesis process of trityl olmesartan medoxomil 浙江华洋药业有限公司 2024-11-29 CN disclosed
CN-119039279-A Synthesis process of trityl olmesartan medoxomil 浙江华洋药业有限公司 2024-11-29 CN disclosed
CN-114835689-B Solvent-free method for preparing irbesartan 浙江金立源药业有限公司 2024-01-02 CN disclosed
CN-115197159-A Preparation method of valsartan intermediate 山东新时代药业有限公司 2022-10-18 CN disclosed
CN-113717118-B Synthesis process of valsartan 安徽美诺华药物化学有限公司 2022-03-01 CN disclosed
CN-113717118-A Synthesis process of valsartan 安徽美诺华药物化学有限公司 2021-11-30 CN disclosed
CN-1082029-A The pyridone that Biphenylmethyl replaces BAYER AG (DE) 1994-02-16 CN disclosed
US-5281604-A Pharmaceuticals AMERICAN CYANAMID COMPANY (US) 1994-01-25 US disclosed
US-5210211-A 4-(1H-PYRROL-1-YL) IMIDAZOLES WITH ANGIOTENSION II ANTAGONIST ACTIVITY WARNER-LAMBERT COMPANY (US) 1993-05-11 US disclosed
CN-1070912-A Imidazopyridine derivatives and preparation method thereof TANABE SEIYAKU CO (JP) 1993-04-14 CN disclosed
WO-1993000341-A1 4-(1-H-PYRROL-1-YL)IMIDAZOLES WITH ANGIOTENSIN II ANTAGONIST ACTIVITY WARNER-LAMBERT COMPANY (US) 1993-01-07 WO disclosed
CN-1048546-A Substituted imidazo-fused 6 unit heterocycle as angiotensin II antagonism medicine MERCK & CO INC (US) 1991-01-16 CN disclosed