SCHEMBL5886728

SCHEMBL5886728

Cc1nc(N2CCN(c3ccc(F)cc3)CC2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTNNB1 P35222 6/20 0.48
TCF7L2 Q9NQB0 6/20 0.48
TP53 P04637 2/20 0.47
LMNA P02545 1/20 0.42
HTR7 P34969 3/20 0.42
MAPT P10636 1/20 0.42
SCD O00767 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5886891 0.95 TP53 (0.44) CTNNB1TCF7L2TP53LMNAHTR7
SCHEMBL5887641 0.92 MAPT (0.44) CTNNB1TCF7L2TP53LMNAHTR7
SCHEMBL5887425 0.92 HTR7 (0.45) CTNNB1TCF7L2TP53LMNAHTR7
SCHEMBL5887548 0.91 KMT2A (0.46) CTNNB1TCF7L2TP53LMNAMAPT
SCHEMBL5887117 0.91 SMN1; SMN2 (0.49) CTNNB1TCF7L2TP53HTR7
SCHEMBL5886779 0.91 MAPT (0.44) CTNNB1TCF7L2TP53LMNAMAPT
SCHEMBL5886882 0.90 MAPT (0.43) TP53LMNAMAPT
SCHEMBL5886707 0.90 ALDH1A1 (0.46) CTNNB1TCF7L2TP53LMNAMAPT
SCHEMBL5887414 0.90 CCR1 (0.43) CTNNB1TCF7L2LMNAMAPT
SCHEMBL5886918 0.90 CTNNB1 (0.43) CTNNB1TCF7L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP CTNNB1 1452/4885TCF7L2 381/4885TP53 43/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.