SCHEMBL5887008

SCHEMBL5887008

Cc1nc(Sc2nc3ccccc3[nH]2)nc2c1ccc(=O)n2-c1ccc(C(N)=O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
HIF1A Q16665 1/20 0.40
CHEK1 O14757 1/20 0.37
LMNA P02545 1/20 0.36
ALDH1A1 P00352 6/20 0.36
MAPT P10636 4/20 0.36
PKM P14618 1/20 0.35
KMT2A Q03164 4/20 0.35
MEN1 O00255 3/20 0.35
HCRTR1 O43613 1/20 0.35
TDP1 Q9NUW8 4/20 0.35
POLB P06746 3/20 0.35
RECQL P46063 1/20 0.35
DUSP3 P51452 1/20 0.35
PTPN5 P54829 1/20 0.35
PTPN11 Q06124 1/20 0.35
CTDSP1 Q9GZU7 1/20 0.35
PDE10A Q9Y233 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887116 0.85 MAPT (0.46) SMN1; SMN2LMNAALDH1A1MAPTKMT2A
SCHEMBL5886826 0.82 POLB (0.41) SMN1; SMN2NPC1RAB9ALMNAALDH1A1
SCHEMBL5886995 0.81 LMNA (0.40) SMN1; SMN2LMNAALDH1A1MAPTRXFP1
SCHEMBL5887005 0.81 TSHR (0.47) SMN1; SMN2ALDH1A1MAPTKMT2AMEN1
SCHEMBL5886758 0.81 LMNA (0.39) NPC1RAB9ALMNAALDH1A1MAPT
SCHEMBL5886939 0.80 RECQL (0.39) SMN1; SMN2NPC1RAB9ALMNAALDH1A1
SCHEMBL5887058 0.78 TSHR (0.34) ALDH1A1KMT2AMEN1KDM4EL3MBTL1
SCHEMBL5887215 0.78 RXRA (0.39) SMN1; SMN2LMNAALDH1A1MAPTKMT2A
SCHEMBL5886741 0.75 LMNA (0.42) SMN1; SMN2NPC1RAB9ALMNAALDH1A1
SCHEMBL5886944 0.69 RXRA (0.47) SMN1; SMN2ALDH1A1MAPTPKMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US claimed
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors PHARMACIA ITALIA S.P.A. 2004-01-15 US claimed
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040009993-A1 Pyridopyrimidinones derivatives as telomerase inhibitors TERT, TERF2, TERF2IP SMN1; SMN2 2219/4885NPC1 4067/4885RAB9A 3217/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.