SCHEMBL5887075

SCHEMBL5887075

CS(=O)(=O)C1=CC[CH]C(c2cccc(Cl)c2)=C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.39
ATM Q13315 1/20 0.37
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
SCD O00767 1/20 0.35
PGR P06401 2/20 0.34
NR3C1 P04150 1/20 0.34
NR3C2 P08235 1/20 0.34
AR P10275 1/20 0.34
PTGS1 P23219 1/20 0.34
HTR2C P28335 2/20 0.33
SLC6A3 Q01959 1/20 0.33
HSD11B1 P28845 1/20 0.33
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4009323 0.81 PTGS2 (0.43) PTGS2PGRPTGS1
SCHEMBL5887567 0.77 CA1 (0.39) PTGS2ATMPTGS1SLC6A3ESR2
SCHEMBL4801089 0.75 NOTUM (0.40) HTR2CSLC6A3
SCHEMBL9650518 0.74 HTR2C (0.37) RAB9AHTR2CESR2
SCHEMBL4014782 0.74 PGR (0.36) PGRHTR2CHTR1AHTR7ESR2
SCHEMBL6407852 0.71 CACNA2D1 (0.38) RAB9AKMT2AHTR2C
SCHEMBL6047625 0.71 HTR2C (0.35) RAB9AKMT2AHTR2CHTR1AHTR7
SCHEMBL16163353 0.69
SCHEMBL15272914 0.69 PTGS2 (0.41) PTGS2PTGS1
SCHEMBL6743237 0.64 PTGS2 (0.38) PTGS2ATMRAB9AKMT2ASCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed
US-20060004195-A1 Alpha,beta-unsaturated esters and acids by stereoselective dehydration JANSSEN PHARMACEUTICA N.V. (BE) 2006-01-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004195-A1 Alpha,beta-unsaturated esters and acids by stereoselective dehydration CCKAR, CCKBR, FFAR1 PTGS2 1436/4885ATM 1914/4885RAB9A 1988/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.