SCHEMBL5887131

SCHEMBL5887131

Cc1nc(N2CC3CC2CN3Cc2ccccc2)nc2c1ccc(=O)n2-c1ccc(C(=O)NCc2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
LMNA P02545 2/20 0.38
HPGD P15428 1/20 0.38
ALOX12 P18054 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PTGER4 P35408 3/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
LTA4H P09960 1/20 0.38
DCTPP1 Q9H773 1/20 0.37
ALDH1A1 P00352 2/20 0.37
PKM P14618 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
OGFRL1 Q5TC84 1/20 0.37
POLB P06746 2/20 0.37
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5887234 0.97 HDAC1 (0.42) HDAC1LMNAHPGDALOX12SMN1; SMN2
SCHEMBL5887537 0.94 ALDH1A1 (0.41) HDAC1LMNAHPGDALOX12SMN1; SMN2
SCHEMBL5887359 0.93 MAOA (0.41) HDAC1LMNAHPGDALOX12SMN1; SMN2
SCHEMBL5887193 0.90 SMN1; SMN2 (0.43) LMNASMN1; SMN2TP53MAPTALDH1A1
SCHEMBL5887463 0.87 LMNA (0.45) HDAC1LMNASMN1; SMN2TP53OPRK1
SCHEMBL5887380 0.87 PPARG (0.41) HDAC1LMNATP53ALDH1A1MEN1
SCHEMBL5887284 0.86 MAPT (0.40) HDAC1LMNATP53MAPTDCTPP1
SCHEMBL5887531 0.86 HDAC1 (0.42) HDAC1LTA4HOPRM1OPRK1
SCHEMBL5887173 0.80 LMNA (0.39) LMNAL3MBTL1PTGER4TP53MAPT
SCHEMBL5887418 0.80 LMNA (0.39) LMNAL3MBTL1TP53MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7019002-B2 Substituted on 8th position with benzoic acid, ester or amide groups; anticancer agents PHARMACIA & UPJOHN, S.P.A. (IT) 2006-03-28 US disclosed