SCHEMBL5887447

SCHEMBL5887447

COc1cc[c]c(-c2cccc(N(C)C)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 7/20 0.46
HSD17B1 P14061 6/20 0.46
FYN P06241 4/20 0.39
MTNR1A P48039 1/20 0.38
MTNR1B P49286 1/20 0.38
NOTUM Q6P988 2/20 0.38
APP P05067 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL323109 0.84 DYRK1A (0.49) NOTUM
SCHEMBL8063028 0.83 APP (0.49) APP
SCHEMBL16719334 0.80 NFE2L2 (0.46)
SCHEMBL7033071 0.79 CA4 (0.43)
SCHEMBL4288060 0.78 HSD17B1 (0.44) HSD17B2HSD17B1FYN
SCHEMBL7101700 0.78 MAOB (0.42)
SCHEMBL10887641 0.76 APP (0.46) APP
SCHEMBL9509841 0.76 TLR9 (0.42) HSD17B2HSD17B1APP
SCHEMBL10918406 0.76 CYP11B1 (0.44)
SCHEMBL11233784 0.76 ALDH1A1 (0.46) FYNNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7037931-B2 Corticotropin releasing factor moderator; analgesics; drug abruse, drug dependency; schizophrenia JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-02 US claimed