SCHEMBL594373

SCHEMBL594373

CC(C)(C)C(=O)Nc1ncc(-c2cccc(C(F)(F)F)c2)s1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
ALDH1A1 P00352 2/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
GSTO1 P78417 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
FFAR2 O15552 1/20 0.47
SCD O00767 2/20 0.46
CCNE1 P24864 1/20 0.46
CDK2 P24941 1/20 0.46
CDK5 Q00535 1/20 0.46
IL2 P60568 1/20 0.45
ACP1 P24666 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
DGAT1 O75907 1/20 0.44
MKNK1 Q9BUB5 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10079021 0.84 KDR (0.53) KDRMEN1KMT2AGSTO1HDAC6
SCHEMBL5051437 0.81 IL2 (0.66) KDRMEN1KMT2AGSTO1HDAC6
SCHEMBL6248559 0.81 KDR (0.71) KDRALDH1A1GSTO1SCDCCNE1
SCHEMBL3176327 0.79 LIMK1 (0.52) KDRKMT2AL3MBTL1GSTO1FFAR2
SCHEMBL3169992 0.76 PIK3CA (0.46) KDRKMT2AGSTO1FFAR2SCD
SCHEMBL4292749 0.76 KDR (0.46) KDRKMT2AGSTO1FFAR2SCD
SCHEMBL21962874 0.73 KDR (0.60) KDRMEN1KMT2AALDH1A1L3MBTL1
SCHEMBL1764981 0.73 ALDH1A1 (0.48) ALDH1A1L3MBTL1HDAC6CDK2CDK5
SCHEMBL2896337 0.72 NR3C1 (0.62) KDRGSTO1FFAR2SCDCCNE1
SCHEMBL12991170 0.72 MEN1 (0.48) KDRMEN1KMT2ACCNE1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-8114993-B2 Use of aryl chlorides in palladium-catalyzed C-H bond functionalization THE UNIVERSITY OF HOUSTON SYSTEM (US) 2012-02-14 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION THE UNIVERSITY OF HOUSTON SYSTEM (US) 2009-01-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090012293-A1 USE OF ARYL CHLORIDES IN PALLADIUM-CATALYZED C-H BOND FUNCTIONALIZATION DBH, DDT, CYCS KDR 2417/4885MEN1 3950/4885KMT2A 1775/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.