SCHEMBL5957049

SCHEMBL5957049

C=CCc1cc(Cl)cc2c1O[C@@H](CO)CO2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.34
CYP3A4 P08684 3/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CA2 P00918 2/20 0.31
CA1 P00915 1/20 0.31
PRKAB2 O43741 2/20 0.31
PRKAG1 P54619 2/20 0.31
PRKAA2 P54646 2/20 0.31
PRKAA1 Q13131 2/20 0.31
PRKAG3 Q9UGI9 2/20 0.31
PRKAG2 Q9UGJ0 2/20 0.31
PRKAB1 Q9Y478 2/20 0.31
POLB P06746 1/20 0.31
PTGDR Q13258 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
CYP1A2 P05177 1/20 0.31
MAPT P10636 1/20 0.31
ITGB2 P05107 1/20 0.30
ICAM1 P05362 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083540 0.78 GABRA1 (0.37) HTR1ACA2
SCHEMBL7083543 0.78 GABRA1 (0.37) HTR1ACA2
SCHEMBL13672070 0.71 MAPT (0.36) HTR1AALDH1A1SMN1; SMN2CA2CA1
SCHEMBL13534191 0.69 HTR1A (0.43) HTR1ASMN1; SMN2CA2CA1PRKAB2
SCHEMBL1119121 0.68 CA2 (0.58) HTR1ASMN1; SMN2CA2CA1PRKAB2
SCHEMBL1044791 0.68 CA2 (0.58) HTR1ASMN1; SMN2CA2CA1PRKAB2
SCHEMBL29444745 0.68 CA2 (0.58) HTR1ASMN1; SMN2CA2CA1PRKAB2
SCHEMBL29444759 0.68 CA2 (0.58) HTR1ASMN1; SMN2CA2CA1PRKAB2
SCHEMBL28709527 0.68 CA2 (0.58) HTR1ASMN1; SMN2CA2CA1PRKAB2
SCHEMBL1119175 0.68 CA2 (0.58) HTR1ASMN1; SMN2CA2CA1PRKAB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1726592-A1 Dioxino derivatives and their use as dopanine agonists Wyeth a Corporation of the State of Delaware (US) 2006-11-29 EP disclosed
EP-1375503-A1 Dioxino derivatives and their use as dopanine agonists Wyeth (US) 2004-01-02 EP disclosed
US-5962465-A BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS AMERICAN HOME PRODUCTS CORPORATION (US) 1999-10-05 US disclosed
US-5756532-A Aminomethyl-2 3 8 9-tetrahydro-7H-1 4-dioxino 2 3-E!-indol-8-ones and derivatives AMERICAN HOME PRODUCTS CORPORATION (US) 1998-05-26 US disclosed
EP-0771800-A2 Dioxino derivatives and their use as dopamine agonists AMERICAN HOME PRODUCTS CORPORATION (US) 1997-05-07 EP disclosed