SCHEMBL5983341

SCHEMBL5983341

CC(C)CCNCc1ccc(Oc2cc(F)ccc2C#N)cc1.CC(C)CCNCc1ccc(Oc2ccc(C#N)c(F)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.39
MAPK1 P28482 2/20 0.39
MITF O75030 1/20 0.39
LMNA P02545 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
GPR35 Q9HC97 1/20 0.39
GPR55 Q9Y2T6 1/20 0.39
XBP1 P17861 1/20 0.39
HTT P42858 1/20 0.39
SLC22A12 Q96S37 6/20 0.39
LTA4H P09960 1/20 0.39
EPHX2 P34913 1/20 0.39
AR P10275 3/20 0.39
CACNA1G O43497 1/20 0.38
CACNA1B Q00975 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 2/20 0.37
FNTA P49354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4806229 0.94 NPSR1 (0.44) NPSR1MAPK1MITFLMNACNR1
SCHEMBL4806912 0.92 CACNA1G (0.40) NPSR1MAPK1MITFLMNACNR1
SCHEMBL14080796 0.74 LPAR1 (0.41) ARFNTAFNTBPGGT1BSLC6A4
SCHEMBL14080782 0.71 KCNJ1 (0.40) SLC22A12LTA4HARTRPV4
SCHEMBL3699384 0.70 OPRM1 (0.45) NPSR1MAPK1MITFLMNACNR1
SCHEMBL8549611 0.68 CYP19A1 (0.49) ARCACNA1GCACNA1BFNTAFNTB
SCHEMBL10535321 0.68 TRPV4 (0.55) SLC22A12ARTRPV4
SCHEMBL28748012 0.68 TRPV4 (0.46) SLC22A12ARTRPV4
SCHEMBL14106705 0.67 LPAR1 (0.47) AR
SCHEMBL3694628 0.67 OPRK1 (0.49) NPSR1MAPK1MAPTKCNH2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1699783-A1 OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2006-09-13 EP disclosed
WO-2005066164-A1 OPIOID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2005-07-21 WO disclosed