SCHEMBL5990705

SCHEMBL5990705

COC(=O)C1CC1c1ccc(O)cc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
CA14 Q9ULX7 2/20 0.36
PDK2 Q15119 1/20 0.36
PDK4 Q16654 1/20 0.36
IDO1 P14902 2/20 0.36
FPR1 P21462 1/20 0.35
FPR2 P25090 1/20 0.35
DEGS1 O15121 1/20 0.35
ACHE P22303 1/20 0.35
TBXAS1 P24557 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15428484 0.87 FPR1 (0.35) CYP3A4CYP1A2CYP2D6TSHRMAPK1
SCHEMBL15548710 0.87 FPR1 (0.35) CYP3A4CYP1A2CYP2D6TSHRMAPK1
SCHEMBL3918513 0.85 CA1 (0.43) CYP3A4CYP1A2TSHRCA12CA1
SCHEMBL15428486 0.84 MAOA (0.47) CA12CA1CA2CA9
SCHEMBL6242073 0.83 FFAR1 (0.43) DEGS1
SCHEMBL5989637 0.77 S1PR1 (0.48) CA2
SCHEMBL16229142 0.76 DEGS1 (0.50) CYP3A4CYP1A2IDO1DEGS1SLC6A4
SCHEMBL1100407 0.76 DEGS1 (0.50) CYP3A4CYP1A2IDO1DEGS1SLC6A4
SCHEMBL15430481 0.76 DEGS1 (0.50) CYP3A4CYP1A2IDO1DEGS1SLC6A4
SCHEMBL15430483 0.76 DEGS1 (0.50) CYP3A4CYP1A2IDO1DEGS1SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060257987-A1 Ppar modulators ELI LILLY AND COMPANY 2006-11-16 US disclosed
EP-1660428-A1 PPAR MODULATORS ELI LILLY AND COMPANY (US) 2006-05-31 EP disclosed
WO-2005019151-A1 PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-03-03 WO disclosed