SCHEMBL6002658

SCHEMBL6002658

CN(c1ccc(Cl)cc1)C1CCN(c2ccc(OC3CCCCO3)cc2)CC1.CN(c1ccc(Cl)cc1)C1CCNCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.40
HTR3E A5X5Y0 2/20 0.36
HTR3B O95264 2/20 0.36
ADRB1 P08588 2/20 0.36
HTR3A P46098 2/20 0.36
HTR3D Q70Z44 2/20 0.36
HTR3C Q8WXA8 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
MAPKAPK2 P49137 4/20 0.35
FFAR1 O14842 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
LSS P48449 1/20 0.33
CYP3A4 P08684 1/20 0.33
FPR2 P25090 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
NPY5R Q15761 1/20 0.32
ACACB O00763 1/20 0.32
ALDH1A1 P00352 2/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2090101 0.94 LSS (0.36) LTA4HFFAR1CRHBPCRHR2LSS
SCHEMBL6001476 0.90 KCNH2 (0.35) FFAR1CRHBPCRHR2LSSCYP3A4
SCHEMBL5534813 0.78 ADRB1 (0.49) LTA4HHTR3EHTR3BADRB1HTR3A
SCHEMBL29656929 0.74 ALDH1A1 (0.45) ALDH1A1
SCHEMBL8663836 0.73 SLC6A4 (0.41) SIGMAR1ALDH1A1
SCHEMBL2092295 0.71 NOS2 (0.44) HTR3AFPR2PROKR1ALDH1A1
SCHEMBL14438088 0.71 FPR2 (0.46) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL2090519 0.70 NPY5R (0.45) HTR3EHTR3BADRB1HTR3AHTR3D
SCHEMBL5541756 0.67 KCNH2 (0.41) ALDH1A1
SCHEMBL3500438 0.66 TNK2 (0.44) NPY5RALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed