SCHEMBL6003969

SCHEMBL6003969

[CH2]C(CCCC)c1c[nH]c(-c2ccccc2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.34
ADORA2A P29274 2/20 0.34
ADORA1 P30542 2/20 0.34
ADORA2B P29275 1/20 0.34
PDE5A O76074 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CYP17A1 P05093 1/20 0.33
GPR84 Q9NQS5 2/20 0.33
CDC7 O00311 1/20 0.33
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
CHUK O15111 1/20 0.33
PDPK1 O15530 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
NTRK1 P04629 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28560027 0.80 DHFR (0.39) ADORA3ADORA2AADORA1ADORA2BCDC7
SCHEMBL28566844 0.76 DHFR (0.40) ADORA3ADORA2AADORA1ADORA2BCDC7
SCHEMBL28913415 0.75 DHFR (0.42) ADORA3ADORA2AADORA1ADORA2BPDPK1
SCHEMBL25403426 0.74 ALDH1A1 (0.38) ADORA3ADORA2AADORA1ADORA2BMAPK1
SCHEMBL4119540 0.73 KDM4E (0.40) TSHRNR1H3
SCHEMBL10529535 0.73 ADORA3 (0.37) ADORA3ADORA2AADORA1PDE5APDE3B
SCHEMBL28559979 0.72 ADORA2A (0.37) ADORA3ADORA2AADORA1ADORA2BPDE5A
SCHEMBL25404388 0.71 L3MBTL1 (0.40) MAPK1TSHR
SCHEMBL27843948 0.71 KCNH2 (0.41) ADORA3ADORA2AADORA1ADORA2BPDE5A
Octane SCHEMBL28114785 0.71 GAA (0.42) ADORA2BPDE5APDE3BPDE3AGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed