Sulfadimethoxine

Sulfadimethoxine

SCHEMBL6006340

C=C(C)C(N)=O.COc1cc(NS(=O)(=O)c2ccc(N)cc2)nc(OC)n1

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

folP

The experimentally established mechanism targets of Sulfadimethoxine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.80
LMNA P02545 2/20 0.80
CYP3A4 P08684 1/20 0.80
HTR6 P50406 1/20 0.80
AKT1 P31749 3/20 0.66
HTT P42858 1/20 0.66
SMN1; SMN2 Q16637 1/20 0.66
KMT2A Q03164 5/20 0.63
POLB P06746 3/20 0.57
CYP2C19 P33261 1/20 0.55
NPSR1 Q6W5P4 1/20 0.54
ALOX12 P18054 1/20 0.54
P2RY1 P47900 1/20 0.54
GFER P55789 1/20 0.53
MAPT P10636 1/20 0.53
HPGD P15428 1/20 0.53
MEN1 O00255 1/20 0.52
CHIA Q9BZP6 1/20 0.52
TP53 P04637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfadimethoxine SCHEMBL29363944 0.90 LMNA (1.00) ALDH1A1LMNACYP3A4HTR6AKT1
Sulfadimethoxine SCHEMBL93845 0.90 LMNA (1.00) ALDH1A1LMNACYP3A4HTR6AKT1
Sulfadimethoxine SCHEMBL2430279 0.89 LMNA (0.97) ALDH1A1LMNACYP3A4HTR6AKT1
Sulfadimethoxine SCHEMBL9486265 0.85 ALDH1A1 (0.90) ALDH1A1LMNACYP3A4HTR6AKT1
Sulfadimethoxine SCHEMBL13372563 0.84 ALDH1A1 (0.76) ALDH1A1LMNACYP3A4HTR6AKT1
SCHEMBL5449670 0.83 ALDH1A1 (0.73) ALDH1A1LMNACYP3A4HTR6AKT1
SCHEMBL10031613 0.83 ALDH1A1 (0.80) ALDH1A1LMNACYP3A4HTR6AKT1
SCHEMBL328330 0.82 ALDH1A1 (0.74) ALDH1A1LMNACYP3A4HTR6AKT1
Sulfadimethoxine SCHEMBL23928724 0.80 ALDH1A1 (0.80) ALDH1A1LMNACYP3A4HTR6AKT1
Sulfadimethoxine SCHEMBL17102809 0.80 LMNA (0.80) ALDH1A1LMNACYP3A4HTR6AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1386935-B1 Dual stimuli-responsive hydrogels and their synthetic methods KOREA INST SCI & TECH (KR) 2006-01-25 EP disclosed
US-6784266-B2 BLOCK POLYMERS HAVING BOTH THERMO- AND PH- RESPONSIVE PROPERTIES NECESSARY FOR DRUG DELIVERY SYSTEMS; COPOLYMERS BASED ON A SULFONAMIDE DERIVATIVE OF STYRENE (PH) AND N-ISOPROPYLACRYLAMIDE (HEAT); SULFA DRUGS KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2004-08-31 US disclosed
US-20040024096-A1 Dual stimuli-responsive hydrogels and their synthetic methods KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2004-02-05 US disclosed
EP-1386935-A1 Dual stimuli-responsive hydrogels and their synthetic methods Korea Institute of Science and Technology (KR) 2004-02-04 EP disclosed