SCHEMBL6007489

SCHEMBL6007489

O=C(O)N1C(c2cccc(F)c2)c2[nH]c3cnccc3c2CC12CC2

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.39
MAPT P10636 1/20 0.38
ESR1 P03372 1/20 0.37
ROCK2 O75116 1/20 0.37
CHUK O15111 1/20 0.35
ABCB1 P08183 6/20 0.35
ABCG2 Q9UNQ0 6/20 0.35
TP53 P04637 2/20 0.33
LMNA P02545 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL999957 0.89 KIF11 (0.38) KIF11MAPTESR1ROCK2CHUK
SCHEMBL998662 0.85 KIF11 (0.39) KIF11MAPTESR1ROCK2TP53
SCHEMBL998181 0.84 KIF11 (0.42) KIF11MAPTESR1ABCB1ABCG2
SCHEMBL998567 0.82 KIF11 (0.40) KIF11MAPTESR1ABCB1ABCG2
SCHEMBL997862 0.78 KIF11 (0.41) KIF11MAPTESR1TP53CYP2D6
SCHEMBL997430 0.76 KIF11 (0.61) KIF11MAPTABCB1ABCG2TP53
SCHEMBL997542 0.76 KIF11 (0.38) KIF11MAPTESR1TP53LMNA
SCHEMBL1000700 0.74 KIF11 (0.53) KIF11MAPTABCB1ABCG2TP53
SCHEMBL999207 0.74 KIF11 (0.38) KIF11ESR1CYP2D6
SCHEMBL1000704 0.74 KIF11 (0.36) KIF11MAPTESR1ABCB1ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637521-A1 NOVEL TRICYCLIC HETEROCYCLE COMPOUND ONO PHARMACEUTICAL CO., LTD. (JP) 2006-03-22 EP disclosed