SCHEMBL6014096

SCHEMBL6014096

CCC(CC)(C(N)=O)c1cccc(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
GAA P10253 2/20 0.41
RIPK1 Q13546 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
C1S P09871 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
SCN5A Q14524 3/20 0.40
SCN9A Q15858 3/20 0.40
HTT P42858 1/20 0.39
KIF11 P52732 1/20 0.39
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5898552 0.82 SCN5A (0.48) PARP1CA1CA2CA5ACA9
SCHEMBL15821917 0.80 CES2 (0.47) ALDH1A1KIF11
SCHEMBL1141842 0.79 OGG1 (0.42) CA1CA2CA5ACA9GAA
SCHEMBL431187 0.78 HTT (0.59) KMT2AALDH1A1HTTKIF11MAPT
SCHEMBL4856143 0.78 PARP1 (0.50) PARP1SMN1; SMN2L3MBTL1KIF11
SCHEMBL16056375 0.77 KMT2A (0.60) PARP1CA1CA2CA5ACA9
SCHEMBL20707128 0.74 ALDH1A1 (0.44) PARP1CA1CA2CA5ACA9
SCHEMBL23326602 0.74 CA1 (0.54) PARP1CA1CA2CA5ACA9
SCHEMBL16183044 0.74 ESR1 (0.40) SMN1; SMN2KMT2AMEN1ALDH1A1HTT
SCHEMBL16081706 0.73 PARP1 (0.44) PARP1CA1CA2CA5ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689229-A1 ARTHROPOD REPELLENT PHARMACOPHORE MODELS, COMPOUNDS IDENTIFIED AS FITTING THE PHARMACOPHORE MODELS, AND METHODS OF MAKING AND USING THEREOF United States Army Medical Research and Materiel Command (US) 2006-08-16 EP disclosed
WO-2005046329-A1 ARTHROPOD REPELLENT PHARMACOPHORE MODELS, COMPOUNDS IDENTIFIED AS FITTING THE PHARMACOPHORE MODELS, AND METHODS OF MAKING AND USING THEREOF UNITED STATES MEDICAL RESEARCH AND MATERIEL COMMAND (US) 2005-05-26 WO disclosed