SCHEMBL6015301

SCHEMBL6015301

C[C](C)C[C@@H]1CCCN(C(N)=O)C1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
MAPK1 P28482 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
LMNA P02545 2/20 0.37
POLB P06746 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SYK P43405 1/20 0.36
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
EPHX2 P34913 2/20 0.35
KDM4E B2RXH2 1/20 0.35
KAT8 Q9H7Z6 1/20 0.35
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
CPN1 P15169 1/20 0.33
CPB2 Q96IY4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15774971 0.86 ITGB3 (0.39) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL14813701 0.82 ALDH1A1 (0.43) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL13548205 0.80 EPHX2 (0.47) ALDH1A1POLBNPC1RAB9ASMN1; SMN2
SCHEMBL1011679 0.80 ITGB3 (0.40) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL28786378 0.80 ITGB3 (0.40) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL24449560 0.79 ALDH1A1 (0.38) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL14813742 0.79 LMNA (0.43) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL29889243 0.78 ALDH1A1 (0.39) ALDH1A1MAPK1LMNAPOLBEPHX2
SCHEMBL1009375 0.77 ITGB3 (0.41) ALDH1A1MAPK1ITGB3ITGA2BLMNA
SCHEMBL15774600 0.74 LTA4H (0.37) ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732920-A2 THIOPHENE DERIVATIVES AS CHK 1 INHIBITORS AstraZeneca AB (SE) 2006-12-20 EP disclosed
WO-2005066163-A2 THIOPHENE DERIVATIVES AS CHK 1 INIHIBITORS ASTRAZENECA AB (SE) 2005-07-21 WO disclosed