SCHEMBL6015537

SCHEMBL6015537

Nc1nc(O)nc2cccc(OC3CCNCC3)c12

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.43
DCPS Q96C86 2/20 0.41
DHFR P00374 1/20 0.41
QPCT Q16769 1/20 0.41
QPCTL Q9NXS2 1/20 0.41
HTR1A P08908 2/20 0.40
SLC6A2 P23975 2/20 0.40
SLC6A3 Q01959 2/20 0.40
KHK P50053 1/20 0.38
ROCK1 Q13464 1/20 0.38
MAP3K5 Q99683 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015554 0.85 DCPS (0.55) DCPSDHFRQPCTQPCTL
SCHEMBL6015541 0.82 DCPS (0.59) DCPSDHFR
SCHEMBL6015546 0.80 DCPS (0.50) DCPSDHFRQPCTQPCTL
SCHEMBL6015540 0.80 DCPS (0.47) DCPSDHFR
SCHEMBL6015552 0.78 DCPS (0.54) DCPSDHFRSLC6A2SLC6A3
SCHEMBL13982644 0.77 HRH1 (0.43) HRH1QPCTQPCTLHTR1ASLC6A2
SCHEMBL15284428 0.74 DCPS (0.59) DCPSDHFR
SCHEMBL6015547 0.73 CHRNB2 (0.51) DCPSDHFR
SCHEMBL6015539 0.73 CHRNB2 (0.51) DCPSDHFR
SCHEMBL15283746 0.73 DCPS (0.57) DCPSDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054526-A2 CHEMOSENSORY RECEPTOR LIGAND-BASED THERAPIES ELCELYX THERAPEUTICS, INC. (US) 2012-04-26 WO disclosed