SCHEMBL6015692

SCHEMBL6015692

CN1CCN(C(C(N)=O)n2c[c]c3cccnc32)CC1

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
PRKCQ Q04759 1/20 0.33
CHIA Q9BZP6 1/20 0.33
CHRM1 P11229 3/20 0.32
ALDH1A1 P00352 2/20 0.32
CHRM5 P08912 1/20 0.32
PARP1 P09874 1/20 0.32
HTR6 P50406 1/20 0.32
SLC1A2 P43004 1/20 0.32
MEN1 O00255 1/20 0.32
TP53 P04637 1/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
ESR2 Q92731 1/20 0.32
IDH1 O75874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27620065 0.80 SIGMAR1 (0.37) CHRM1CHRM5MEN1KMT2A
SCHEMBL7832110 0.70 PDE4A (0.35)
SCHEMBL5802988 0.68 PARP1 (0.53) PARP1
SCHEMBL6015693 0.68 ALDH1A1 (0.41) CHIAALDH1A1TP53HTT
SCHEMBL6015675 0.67 TDP1 (0.46) CHRM1MEN1KMT2A
SCHEMBL30499312 0.65 IDH1 (0.49) ALDH1A1SLC1A2TP53ALOX12HTT
SCHEMBL2980811 0.65 FEN1 (0.34)
SCHEMBL30499284 0.62 KCNA5 (0.46) CHRM1ALDH1A1HTTIDH1
SCHEMBL1561088 0.62 POLB (0.44) PARP1
SCHEMBL3641753 0.62 SLC1A2 (0.62) CHRM1ALDH1A1SLC1A2MEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed