SCHEMBL6015693

SCHEMBL6015693

CN1CCN(NC(=O)Cn2c[c]c3cccnc32)CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
CHIA Q9BZP6 1/20 0.37
MAPT P10636 3/20 0.36
GAA P10253 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
ACHE P22303 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015665 0.82 OPRK1 (0.48) ALDH1A1TP53
SCHEMBL6015675 0.79 TDP1 (0.46)
SCHEMBL6015666 0.75 PTGS2 (0.38) ALDH1A1TP53MAPTHDAC6
SCHEMBL6015933 0.71 HSD11B1 (0.43) ALDH1A1GAA
SCHEMBL6015925 0.71 TSHR (0.54) ALDH1A1TP53MAPTCYP2C19CYP3A4
SCHEMBL6015802 0.71 MEN1 (0.46) ALDH1A1TP53HTTMAPTHPGD
SCHEMBL6015703 0.71 REN (0.39)
SCHEMBL6016000 0.69 CYP1A2 (0.33) ALDH1A1HTTGAA
SCHEMBL6015692 0.68 HRH4 (0.33) ALDH1A1TP53HTTCHIA
SCHEMBL6015787 0.66 CBX7 (0.44) ALDH1A1MAPTGAACYP2C19HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP disclosed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO disclosed