SCHEMBL6016470

SCHEMBL6016470

N#CCc1ncc(C(=O)O)c(-c2ccccc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.42
LMNA P02545 4/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAPK1 P28482 1/20 0.42
ATM Q13315 1/20 0.42
MEN1 O00255 6/20 0.42
KMT2A Q03164 6/20 0.42
KDM4E B2RXH2 2/20 0.42
POLB P06746 1/20 0.42
LDHA P00338 1/20 0.39
HPGD P15428 1/20 0.39
THRB P10828 1/20 0.38
CYP1A2 P05177 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
ATR Q13535 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016363 0.82 LMNA (0.46) NTRK1LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL17111548 0.80 NTRK1 (0.52) NTRK1
SCHEMBL27488851 0.78 LMNA (0.43) LMNAALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL6016399 0.78 ALDH1A1 (0.49) LMNAALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL6016349 0.78 NTRK1 (0.45) NTRK1LMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL18779324 0.78 JAK2 (0.44) NTRK1LMNAALDH1A1MAPTMEN1
SCHEMBL6016450 0.77 MEN1 (0.51) LMNAALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL8399319 0.73 MEN1 (0.49) LMNAALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL6016478 0.73 MEN1 (0.69) LMNAALDH1A1MAPTSMN1; SMN2MAPK1
SCHEMBL7709570 0.73 TAAR1 (0.47) LMNAALDH1A1MAPTSMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed
EP-1187815-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed
WO-2000073279-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed