SCHEMBL6016399

SCHEMBL6016399

CCCc1ncc(C(=O)O)c(-c2ccccc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
MAPT P10636 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 2/20 0.49
MAPK1 P28482 1/20 0.49
ATM Q13315 1/20 0.49
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
AGTR1 P30556 2/20 0.44
AGTR2 P50052 2/20 0.44
KDM4E B2RXH2 3/20 0.43
LDHA P00338 1/20 0.43
HPGD P15428 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
GPR84 Q9NQS5 1/20 0.42
PKM P14618 1/20 0.42
HSD17B10 Q99714 1/20 0.42
THRB P10828 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016363 0.83 LMNA (0.46) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL6016450 0.81 MEN1 (0.51) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL27488851 0.79 LMNA (0.43) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL6016349 0.79 NTRK1 (0.45) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL6016470 0.78 NTRK1 (0.42) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL31324954 0.76 GABRP (0.42) ALDH1A1MAPTSMN1; SMN2LMNAMEN1
SCHEMBL400143 0.76 NTRK1 (0.60) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL6016324 0.75 CHRM5 (0.46) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL6016466 0.75 CYP11B1 (0.51)
SCHEMBL8399319 0.74 MEN1 (0.49) ALDH1A1MAPTSMN1; SMN2LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed
EP-1187815-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed
WO-2000073279-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed