SCHEMBL6017387

SCHEMBL6017387

CCOC(=O)Cc1c[nH]c2ccc(OCc3cnc(-c4ccc(C(F)(F)F)cc4)nc3C3CC3)cc12

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.40
MAOB P27338 1/20 0.40
PKM P14618 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.38
ICMT O60725 2/20 0.37
HCRTR2 O43614 1/20 0.36
PPARD Q03181 3/20 0.36
PPARA Q07869 2/20 0.36
GSTP1 P09211 2/20 0.36
PPARG P37231 1/20 0.36
IGF1R P08069 1/20 0.36
MET P08581 1/20 0.36
SRC P12931 1/20 0.36
LTA4H P09960 1/20 0.35
PLA2G2A P14555 1/20 0.35
SCN9A Q15858 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017580 0.94 MAOB (0.40) TRPV1MAOBPKMPPARDPPARA
SCHEMBL6017240 0.90 KDM4E (0.43) TRPV1ICMTPPARDPPARAPPARG
SCHEMBL6017371 0.89 TRPV1 (0.45) TRPV1MAOBPKMTRPM8ICMT
SCHEMBL6017230 0.87 PKM (0.38) TRPV1MAOBPKMPPARDPPARA
SCHEMBL6017575 0.85 TRPV1 (0.46) TRPV1MAOBPKMTRPM8ICMT
SCHEMBL5617383 0.84 PPARD (0.43) MAOBPPARDPPARAPPARG
SCHEMBL1550166 0.81 PPARD (0.49) MAOBPPARDPPARAGSTP1PPARG
SCHEMBL5617133 0.80 KDM4E (0.48) TRPV1ICMTPPARDPPARAPPARG
SCHEMBL6030172 0.79 PPARD (0.44) MAOBPPARDPPARAGSTP1
SCHEMBL6029336 0.78 PPARD (0.51) MAOBPPARDPPARAGSTP1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed