SCHEMBL6017580

SCHEMBL6017580

CCOC(=O)Cc1c[nH]c2cc(OCc3cnc(-c4ccc(C(F)(F)F)cc4)nc3C3CC3)ccc12

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.40
PKM P14618 1/20 0.39
PPARD Q03181 7/20 0.37
PPARA Q07869 6/20 0.37
GSTP1 P09211 3/20 0.36
IGF1R P08069 1/20 0.34
MET P08581 1/20 0.34
SRC P12931 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
FOS P01100 1/20 0.34
JUN P05412 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
TRPV1 Q8NER1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017387 0.94 TRPV1 (0.40) MAOBPKMPPARDPPARAGSTP1
SCHEMBL6017230 0.93 PKM (0.38) MAOBPKMPPARDPPARAGSTP1
SCHEMBL5617383 0.90 PPARD (0.43) MAOBPPARDPPARA
SCHEMBL6017240 0.84 KDM4E (0.43) PPARDPPARANFKB1TRPV1
SCHEMBL6017141 0.83 PPARA (0.39) PPARDPPARATRPV1
SCHEMBL6017371 0.83 TRPV1 (0.45) MAOBPKMPPARDPPARAGSTP1
SCHEMBL6017361 0.81 PKM (0.42) MAOBPKMPPARDPPARAIGF1R
SCHEMBL1550166 0.81 PPARD (0.49) MAOBPPARDPPARAGSTP1
SCHEMBL6017372 0.80 PKM (0.43) MAOBPKMPPARDPPARAIGF1R
SCHEMBL6017575 0.79 TRPV1 (0.46) MAOBPKMPPARDPPARAGSTP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed