SCHEMBL6017265

SCHEMBL6017265

CCOC(=O)Cc1c[nH]c2cc(OCc3ccc(-c4ccc(OC(F)(F)F)cc4)nc3C(F)(F)F)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
PPARD Q03181 3/20 0.39
MAPT P10636 4/20 0.38
PTGER4 P35408 1/20 0.37
PRMT5 O14744 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 2/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
POLB P06746 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
GSK3B P49841 1/20 0.35
LMNA P02545 1/20 0.35
AHR P35869 1/20 0.35
MAT2A P31153 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
ICMT O60725 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5653757 0.89 PPARD (0.41) PPARDPTGER4KDM4EALDH1A1HPGD
SCHEMBL6017359 0.85 PKM (0.42) PKMPPARDMAPTPTGER4ALDH1A1
SCHEMBL6017372 0.85 PKM (0.43) PKMPPARDPRMT5TRPV1
SCHEMBL6065143 0.82 PKM (0.42) PKMPPARDMAPTPTGER4ALDH1A1
SCHEMBL6017323 0.81 PKM (0.45) PKMPPARDMAPTPRMT5KDM4E
SCHEMBL9662589 0.80 PKM (0.60) PKMMAPTKDM4EALDH1A1POLB
SCHEMBL6064759 0.80 PKM (0.40) PKMPPARDMAPTPTGER4PRMT5
SCHEMBL6065162 0.80 PKM (0.40) PKMPPARDMAPTPTGER4ALDH1A1
SCHEMBL6017361 0.78 PKM (0.42) PKMPPARDMAPT
SCHEMBL6065368 0.78 PKM (0.41) PKMMAPTALDH1A1HPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed