SCHEMBL6017323

SCHEMBL6017323

CCOC(=O)Cc1c[nH]c2cc(OCc3ccc(-c4cccc(C(F)(F)F)c4)nc3C)ccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.45
GRIN1 Q05586 2/20 0.41
GRIN2B Q13224 2/20 0.41
MAPT P10636 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
IGF1R P08069 2/20 0.38
MET P08581 2/20 0.38
SRC P12931 2/20 0.38
ICMT O60725 1/20 0.38
SSTR1 P30872 1/20 0.38
SSTR3 P32745 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
TRPM8 Q7Z2W7 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
KMO O15229 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017372 0.93 PKM (0.43) PKMIGF1RMETSRCPPARD
SCHEMBL5617387 0.83 PPARD (0.49) PPARDPPARA
SCHEMBL6017265 0.81 PKM (0.42) PKMMAPTMEN1KMT2AICMT
SCHEMBL6017227 0.81 PKM (0.41) PKMMAPTMEN1KMT2AKDM4E
SCHEMBL6017361 0.79 PKM (0.42) PKMMAPTIGF1RMETSRC
SCHEMBL6028284 0.77 GRIN2B (0.47) GRIN1GRIN2BMAPTMEN1KMT2A
SCHEMBL6064609 0.76 PKM (0.42) PKMMAPTPPARDPPARAMAOB
SCHEMBL5617384 0.76 PPARD (0.45) KDM4EPPARDPPARA
SCHEMBL6017371 0.75 TRPV1 (0.45) PKMIGF1RMETSRCICMT
SCHEMBL6017580 0.75 MAOB (0.40) PKMIGF1RMETSRCPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed