SCHEMBL6017575

SCHEMBL6017575

CCOC(=O)Cc1c[nH]c2ccc(OCc3cnc(-c4ccc(C(F)(F)F)cc4)nc3CCOC)cc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 6/20 0.46
HCRTR2 O43614 1/20 0.42
MAOB P27338 1/20 0.40
TRPM8 Q7Z2W7 1/20 0.39
PKM P14618 1/20 0.39
PPARD Q03181 2/20 0.38
PPARG P37231 1/20 0.38
PPARA Q07869 1/20 0.38
GSTP1 P09211 1/20 0.38
ICMT O60725 2/20 0.37
LTA4H P09960 2/20 0.37
PLA2G2A P14555 2/20 0.37
IGF1R P08069 1/20 0.37
MET P08581 1/20 0.37
SRC P12931 1/20 0.37
USP2 O75604 1/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017333 0.91 TRPV1 (0.48) TRPV1HCRTR2PPARDPPARGPPARA
SCHEMBL6017371 0.89 TRPV1 (0.45) TRPV1HCRTR2MAOBTRPM8PKM
SCHEMBL6017118 0.85 PKM (0.38) TRPV1MAOBTRPM8PKMPPARD
SCHEMBL6017387 0.85 TRPV1 (0.40) TRPV1HCRTR2MAOBTRPM8PKM
SCHEMBL5617133 0.80 KDM4E (0.48) TRPV1PPARDPPARGPPARAICMT
SCHEMBL6218951 0.79 PPARG (0.51) PPARDPPARGPPARA
SCHEMBL6017580 0.79 MAOB (0.40) TRPV1MAOBPKMPPARDPPARA
SCHEMBL6219446 0.79 PPARA (0.59) PPARDPPARGPPARA
SCHEMBL6029277 0.78 PPARD (0.51) MAOBPPARDPPARGPPARAGSTP1
SCHEMBL6220042 0.78 PPARD (0.49) TRPV1TRPM8PKMPPARDPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed