SCHEMBL60190

SCHEMBL60190

CNc1nc(N)nc(N(C)C)n1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
HSD17B10 Q99714 2/20 0.42
CYP1A2 P05177 1/20 0.42
THRB P10828 1/20 0.42
BLM P54132 1/20 0.42
CREBBP Q92793 1/20 0.42
PDE4A P27815 1/20 0.41
NUDT1 P36639 1/20 0.41
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
TSHR P16473 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 4/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
AHR P35869 1/20 0.35
RAB9A P51151 1/20 0.35
KDM4E B2RXH2 2/20 0.34
GAA P10253 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32675859 1.00 LMNA (0.42) LMNAHSD17B10CYP1A2THRBBLM
Methylamine SCHEMBL17309971 0.96 PDE4A (0.40) LMNAHSD17B10CYP1A2THRBBLM
Formaldehyde SCHEMBL6476807 0.94 POLB (0.40) LMNAHSD17B10CYP1A2THRBBLM
Altretamine SCHEMBL1978783 0.91 LMNA (0.48) LMNAHSD17B10CYP1A2THRBBLM
Acetic Acid SCHEMBL28195268 0.89 POLB (0.49) LMNAHSD17B10CYP1A2THRBBLM
SCHEMBL19144867 0.88 CA1 (0.40) LMNAHSD17B10CYP1A2THRBBLM
SCHEMBL1033226 0.84 CYP1A2 (0.53) LMNAHSD17B10CYP1A2THRBBLM
Pentamethyl Melamine SCHEMBL38832 0.84 LMNA (0.61) LMNAHSD17B10CYP1A2THRBBLM
Altretamine SCHEMBL4448907 0.84 LMNA (0.61) LMNAHSD17B10CYP1A2THRBBLM
Pentamethyl Melamine SCHEMBL15346326 0.81 LMNA (0.58) LMNAHSD17B10CYP1A2THRBBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1889 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12364682-B2 Use of tegaserod in preparation of anti-tumor drug QINGDAO HAIJI BIOMEDICINE CO., LTD. (CN) 2025-07-22 US claimed
US-20250059301-A1 Fusion Protein Construct NORTHWESTERN UNIVERSITY 2025-02-20 US claimed
CN-119463251-A PVA/PEO/PU composite water-soluble patterned film and preparation method and application thereof 孙琇芳 2025-02-18 CN claimed
US-20240316079-A1 USE OF AKR1C3-ACTIVATED COMPOUND OBI PHARMA, INC. (CN) 2024-09-26 US claimed
CN-118105513-A Conjugates comprising self-degrading groups and methods related thereto 乐高化学生物科学股份有限公司 2024-05-31 CN claimed
CN-118046691-A Acrylic acid type water-soluble pattern film, preparation method and application thereof 孙琇芳 2024-05-17 CN claimed
EP-4297872-A1 USE OF AKR1C3-ACTIVATED COMPOUND OBI Pharma, Inc. (TW) 2024-01-03 EP claimed
CN-117244076-A Conjugates comprising self-degrading groups and methods related thereto 乐高化学生物科学股份有限公司 2023-12-19 CN claimed
CN-116999571-A Antibody-drug conjugates comprising anti-B7-H3 antibodies 尹图赛利有限公司 2023-11-07 CN claimed
CN-113929930-B Temperature-responsive persulfate slow-release gel and preparation method and application thereof 中国环境科学研究院 2023-08-11 CN claimed
US-20040023961-A1 Aryl ureas with raf kinase and angiogenisis inhibiting activity BAYER CORPORATION 2004-02-05 US claimed
US-20030216396-A1 Pyridine, quinoline, and isoquinoline N-oxides as kinase inhibitors BAYER CORPORATION 2003-11-20 US claimed
US-20030216446-A1 Aryl ureas as kinase inhibitors BAYER CORPORATION (US) 2003-11-20 US claimed
WO-2003068223-A1 ARYL UREAS WITH RAF KINASE AND ANGIOGENESIS INHIBITING ACTIVITY BAYER CORPORATION (US) 2003-08-21 WO claimed
WO-2003068746-A1 ARYL UREAS AS KINASE INHIBITORS BAYER PHARMACEUTICALS CORPORATION (US) 2003-08-21 WO claimed
WO-2003055890-A1 THIENOPYRIMIDINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO claimed
WO-2003055489-A1 2,4-DIAMINO-PYRIMIDINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO claimed
WO-2003055866-A1 QUINAZOLINE AND QUINOLINE DERIVATIVE COMPOUNDS AS INHIBITORS OF PROLYLPEPTIDASE, INDUCERS OF APOPTOSIS AND CANCER TREATMENT AGENTS BAYER PHARMACEUTICALS CORPORATION (US) 2003-07-10 WO claimed
WO-2003040141-A1 OXAZOLYL-PHENYL-2,4-DIAMINO-PYRIMIDINE COMPOUNDS AND METHODS FOR TREATING HYPERPROLIFERATIVE DISORDERS BAYER PHARMACEUTICALS CORPORATION (US) 2003-05-15 WO claimed
US-5534625-A 2,4,6-TRIAMINO-1,3,5-TRIAZINE DERIVATIVES; OVARIES CANCER RESEARCH TECHNOLOGY LIMITED (GB) 1996-07-09 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12364682-B2 Use of tegaserod in preparation of anti-tumor drug STAT3, JAK2, JAK1 LMNA 4823/4885HSD17B10 4096/4885CYP1A2 4546/4885
US-20240316079-A1 USE OF AKR1C3-ACTIVATED COMPOUND AKR1A1, AKR1C1, AK1 LMNA 3534/4885HSD17B10 134/4885CYP1A2 641/4885
US-20250059301-A1 Fusion Protein Construct RPS27A, CD2BP2, JMJD7 LMNA 4363/4885HSD17B10 2317/4885CYP1A2 2913/4885
US-20030216396-A1 Pyridine, quinoline, and isoquinoline N-oxides as kinase inhibitors MAP2K2, MAP2K7, MAPK1 LMNA 4406/4885HSD17B10 4542/4885CYP1A2 481/4885
US-20030216446-A1 Aryl ureas as kinase inhibitors MAPK1, MAP3K1, MAP3K6 LMNA 4377/4885HSD17B10 4000/4885CYP1A2 894/4885
US-20040023961-A1 Aryl ureas with raf kinase and angiogenisis inhibiting activity BRAF, FLT1, RAF1 LMNA 4417/4885HSD17B10 4286/4885CYP1A2 2073/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.