SCHEMBL6019499

SCHEMBL6019499

On1c(C(F)(F)F)nc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
KDM4E B2RXH2 2/20 0.54
HPGD P15428 1/20 0.54
LMNA P02545 4/20 0.52
TSHR P16473 1/20 0.52
CYP2C9 P11712 3/20 0.51
CYP2C19 P33261 3/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 1/20 0.51
TP53 P04637 1/20 0.51
MAPK1 P28482 1/20 0.50
CYP3A4 P08684 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PIK3CB P42338 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
MAPT P10636 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11880401 0.81 ALDH1A1 (0.41) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL2958001 0.78 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL10457804 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL1663643 0.77 NOS2 (0.55) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL5851401 0.77 SMN1; SMN2 (0.55) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL5851398 0.77 ALDH1A1 (0.54) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL30034162 0.77 SMN1; SMN2 (0.55) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL3968510 0.77 CYP2C9 (0.62) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL12937256 0.76 MAPK1 (0.74) ALDH1A1KDM4EHPGDLMNATSHR
SCHEMBL17378596 0.74 MAPK1 (0.59) ALDH1A1KDM4EHPGDLMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613626-A1 CYCLIC BENZIMIDAZOLES ALTANA Pharma AG (DE) 2006-01-11 EP disclosed
WO-2004087701-A1 CYCLIC BENZIMIDAZOLES ALTANA PHARMA AG (DE) 2004-10-14 WO disclosed
US-4031107-A Method for introducing amino groups into benzimidazole or imidazopyridine compounds ELI LILLY AND COMPANY (US) 1977-06-21 US disclosed